SCHEMBL9056734

SCHEMBL9056734

O=C(O)CCc1ccc(-c2nnc(-c3ccc4c(c3)CCNCC4)s2)cc1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
RXRA P19793 1/20 0.44
RXRB P28702 1/20 0.44
RXRG P48443 1/20 0.44
S1PR1 P21453 14/20 0.43
ITGB3 P05106 1/20 0.41
ITGA2B P08514 1/20 0.41
FFAR1 O14842 2/20 0.41
LMNA P02545 1/20 0.41
FFAR4 Q5NUL3 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9055061 0.85 S1PR1 (0.48) RXRARXRBRXRGS1PR1
Hydrochloric Acid SCHEMBL20509927 0.79 RXRA (0.50) RXRARXRBRXRGITGB3ITGA2B
SCHEMBL9056558 0.76 RXRA (0.42) RXRARXRBRXRGITGB3ITGA2B
SCHEMBL20510025 0.72 PLAU (0.53) RXRARXRBRXRGITGB3ITGA2B
SCHEMBL8560143 0.72 RXRA (0.40) RXRARXRBRXRGITGB3ITGA2B
Hydrochloric Acid SCHEMBL8564229 0.71 MAPK9 (0.38) RXRARXRBRXRGITGB3ITGA2B
SCHEMBL9053431 0.71 LMNA (0.38) LMNAFFAR4
SCHEMBL9053277 0.71 LMNA (0.43) RXRARXRBRXRGLMNAFFAR4
SCHEMBL9058459 0.71 DVL1 (0.39)
SCHEMBL9053434 0.71 EIF4E (0.39) LMNAFFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1996004271-A1 CONDENSED AZEPINE DERIVATIVES, DRUGS CONTAINING THESE COMPOUNDS AND METHODS FOR PREPARING THEM DR. KARL THOMAE GMBH (DE) 1996-02-15 WO disclosed