Methylephedrine

Methylephedrine

SCHEMBL907677

CC([C@@H](O)c1ccccc1)N(C)C

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 1.00
ALDH1A1 P00352 2/20 1.00
AOC3 Q16853 5/20 0.70
GAA P10253 1/20 0.56
ADRA2C P18825 2/20 0.56
ADRA2A P08913 1/20 0.56
LMNA P02545 1/20 0.56
HIF1A Q16665 1/20 0.56
CHRM2 P08172 1/20 0.52
ADRA1A P35348 1/20 0.52
RGS12 O14924 1/20 0.52
GLA P06280 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
PKM P14618 1/20 0.52
ALOX15 P16050 1/20 0.52
TSHR P16473 1/20 0.52
ALOX12 P18054 1/20 0.52
NFKB1 P19838 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Methylephedrine SCHEMBL99674 1.00 KDM4E (1.00) KDM4EALDH1A1AOC3GAAADRA2C
Methylephedrine SCHEMBL907777 1.00 KDM4E (1.00) KDM4EALDH1A1AOC3GAAADRA2C
Methylephedrine SCHEMBL7496690 1.00 KDM4E (1.00) KDM4EALDH1A1AOC3GAAADRA2C
Methylephedrine SCHEMBL338479 1.00 KDM4E (1.00) KDM4EALDH1A1AOC3GAAADRA2C
Methylephedrine SCHEMBL2712293 1.00 KDM4E (1.00) KDM4EALDH1A1AOC3GAAADRA2C
Methylephedrine SCHEMBL11959977 1.00 KDM4E (1.00) KDM4EALDH1A1AOC3GAAADRA2C
Methylephedrine SCHEMBL338478 1.00 KDM4E (1.00) KDM4EALDH1A1AOC3GAAADRA2C
Methylephedrine SCHEMBL99673 1.00 KDM4E (1.00) KDM4EALDH1A1AOC3GAAADRA2C
Methylephedrine SCHEMBL8083321 0.98 KDM4E (0.96) KDM4EALDH1A1AOC3GAAADRA2C
Methylephedrine SCHEMBL68363 0.98 ALDH1A1 (0.96) KDM4EALDH1A1AOC3GAAADRA2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 17 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1314333-A Method for asymmetrically synthesizing secondary propiolic alcohol compound SHANGHAI INST ORGANIC CHEM (CN) 2001-09-26 CN claimed
WO-2019113312-A1 ANTICANCER COMPOUND PROCESS INNOCRIN PHARMACEUTICALS, INC. (US) 2019-06-13 WO disclosed
CN-105164131-A Tricyclic heterocycles as bet protein inhibitors INCYTE CORP 2015-12-16 CN disclosed
CN-102203068-B Cyclohexane derivative and pharmaceutical use thereof TORAY INDUSTRIES 2014-03-19 CN disclosed
CN-102906169-A Nanoporous foaming formulations containing active ingredients based on pharmaceutically acceptable thermoplastically processable polymers BASF SE 2013-01-30 CN disclosed
US-8288569-B2 Carbonyl asymmetric alkylation SANDOZ AG (CH) 2012-10-16 US disclosed
CN-102203068-A Cyclohexane derivative and pharmaceutical use thereof TORAY INDUSTRIES 2011-09-28 CN disclosed
EP-1966127-B1 CARBONYL ASYMMETRIC ALKYLATION SANDOZ AG (CH) 2011-04-06 EP disclosed
US-20110009648-A1 Carbonyl Asymmetric Alkylation SANDOZ AG (CH) 2011-01-13 US disclosed
CN-100582092-C Process for preparing diphenyl azetidinone derivatives AVENTIS PHARMA GMBH 2010-01-20 CN disclosed
EP-1966127-A1 CARBONYL ASYMMETRIC ALKYLATION Sandoz AG (CH) 2008-09-10 EP disclosed
WO-2007082771-A1 CARBONYL ASYMMETRIC ALKYLATION SANDOZ AG (CH) 2007-07-26 WO disclosed
CN-1956951-A Method for producing diphenyl azetidinone derivatives AVENTIS PHARMA GMBH (DE) 2007-05-02 CN disclosed
CN-1197836-C Method for asymmetrically synthesizing secondary propiolic alcohol compound SHANGHAI INST ORGANIC CHEM (CN) 2005-04-20 CN disclosed
CN-1112355-C Difluore methane-sulfonic acid metal reagent, and its synthetic method and use SHANGHAI INST ORGANIC CHEM (CN) 2003-06-25 CN disclosed
CN-1314344-A Difluore methane-sulfonic acid metal reagent, and its synthetic method and use SHANGHAI INST ORGANIC CHEM (CN) 2001-09-26 CN disclosed
CN-1314333-A Method for asymmetrically synthesizing secondary propiolic alcohol compound SHANGHAI INST ORGANIC CHEM (CN) 2001-09-26 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110009648-A1 Carbonyl Asymmetric Alkylation COASY, ADH5, SI KDM4E 880/4885ALDH1A1 53/4885AOC3 345/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.