SCHEMBL9108244

SCHEMBL9108244

Fc1cc(F)c(Br)c(Cl)c1

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 4/20 0.34
KDM1B Q8NB78 3/20 0.34
ALOX15 P16050 1/20 0.32
MAPK14 Q16539 1/20 0.30
CES2 O00748 1/20 0.30
CES1 P23141 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30350420 1.00 KDM1A (0.34) KDM1AKDM1BALOX15MAPK14CES2
SCHEMBL7950256 0.86 IDO1 (0.32) ALOX15
SCHEMBL919665 0.80 KDM1A (0.42) KDM1AKDM1BCES2CES1
SCHEMBL793988 0.79 NMT1 (0.38) KDM1AKDM1B
SCHEMBL28965365 0.79 ALDH1A1 (0.41) KDM1AKDM1BALOX15MAPK14
SCHEMBL6553272 0.77 KDM1A (0.41) KDM1AKDM1BCES2CES1
SCHEMBL1806961 0.75 CYP3A4 (0.46) KDM1AKDM1B
SCHEMBL15287359 0.75 EPAS1 (0.33) ALOX15
SCHEMBL21979280 0.75 CA9 (0.36) ALOX15
SCHEMBL13550170 0.75 RAPGEF4 (0.32)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 81 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250092024-A1 SUBSTITUTED CYCLOHEXYL COMPOUNDS AS NOP INHIBITORS DART NEUROSCIENCE LLC 2025-03-20 US disclosed
US-20250043059-A1 POLYURETHANE ADHESIVE DOW GLOBAL TECHNOLOGIES LLC (US) 2025-02-06 US disclosed
WO-2024175907-A1 MACROCYCLIC ALPHA4BETA7 INTEGRIN INHIBITORS C4X DISCOVERY LIMITED (GB) 2024-08-29 WO disclosed
EP-3681928-B1 PROCESS OF MANUFACTURING POLYOLS DOW GLOBAL TECHNOLOGIES LLC (US) 2024-05-01 EP disclosed
EP-3681928-B1 PROCESS OF MANUFACTURING POLYOLS DOW GLOBAL TECHNOLOGIES LLC (US) 2024-05-01 EP disclosed
US-11970574-B2 Process of manufacturing surfactants and lubricants DOW GLOBAL TECHNOLOGIES LLC (US) 2024-04-30 US disclosed
EP-3681931-B1 PROCESS OF MANUFACTURING SURFACTANTS AND LUBRICANTS DOW GLOBAL TECHNOLOGIES LLC (US) 2024-04-24 EP disclosed
EP-3681930-B1 PROCESS OF MANUFACTURING POLYOLS DOW GLOBAL TECHNOLOGIES LLC (US) 2024-04-24 EP disclosed
US-11958936-B2 Process of manufacturing polyols DOW GLOBAL TECHNOLOGIES LLC (US) 2024-04-16 US disclosed
US-11945808-B2 Substituted cyclohexyl compounds as NOP inhibitors DART NEUROSCIENCE, LLC (US) 2024-04-02 US disclosed
US-9216996-B2 Substituted 2,3,4,5,7,9,13,13a-octahydropyrido[1′,2′:4,5]pyrazino[2,1-b][1,3]oxazepines and methods for treating viral infections GILEAD SCIENCES, INC. (US) 2015-12-22 US disclosed
EP-2822954-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE Gilead Sciences, Inc. (US) 2015-01-14 EP disclosed
US-8853242-B2 Nitrogenous-ring acylguanidine derivative ASTELLAS PHARMA INC. (JP) 2014-10-07 US disclosed
US-20140221356-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2014-08-07 US disclosed
US-20140221356-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2014-08-07 US disclosed
US-20140221356-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. 2014-08-07 US disclosed
WO-2014100323-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE GILEAD SCIENCES, INC. (US) 2014-06-26 WO disclosed
EP-2463276-B1 NITROGENOUS-RING ACYLGUANIDINE DERIVATIVE ASTELLAS PHARMA INC (JP) 2014-03-12 EP disclosed
EP-2463276-A1 NITROGENOUS-RING ACYLGUANIDINE DERIVATIVE Astellas Pharma Inc. (JP) 2012-06-13 EP disclosed
US-20120142727-A1 NITROGENOUS-RING ACYLGUANIDINE DERIVATIVE ASTELLAS PHARMA INC. (JP) 2012-06-07 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11945808-B2 Substituted cyclohexyl compounds as NOP inhibitors OPRL1, OPRK1, NOP56 KDM1A 4230/4885KDM1B 4674/4885ALOX15 3104/4885
US-11970574-B2 Process of manufacturing surfactants and lubricants F12, MSR1, LPAR3 KDM1A 1772/4885KDM1B 1785/4885ALOX15 1181/4885
US-20250092024-A1 SUBSTITUTED CYCLOHEXYL COMPOUNDS AS NOP INHIBITORS OPRL1, OPRK1, NOP56 KDM1A 4230/4885KDM1B 4674/4885ALOX15 3104/4885
US-20250043059-A1 POLYURETHANE ADHESIVE ITGA1, AFF1, PBRM1 KDM1A 186/4885KDM1B 338/4885ALOX15 1094/4885
US-20120142727-A1 NITROGENOUS-RING ACYLGUANIDINE DERIVATIVE HTR5A, HTR2A, HTR1E KDM1A 1737/4885KDM1B 2042/4885ALOX15 1101/4885
US-20140221356-A1 POLYCYCLIC-CARBAMOYLPYRIDONE COMPOUNDS AND THEIR PHARMACEUTICAL USE ZC3HAV1, PYM1, ZC3HAV1L KDM1A 510/4885KDM1B 756/4885ALOX15 3518/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.