SCHEMBL9119858

SCHEMBL9119858

Cc1ccoc2c(N3CCNCC3)ccc1-2

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 2/20 0.51
ADRB1 P08588 2/20 0.49
HTR3A P46098 5/20 0.45
HTR3E A5X5Y0 1/20 0.45
HTR3B O95264 1/20 0.45
HTR3D Q70Z44 1/20 0.45
HTR3C Q8WXA8 1/20 0.45
HTR1A P08908 4/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9119205 0.83 ADRB1 (0.49) HTR7ADRB1HTR3AHTR3EHTR3B
SCHEMBL9119128 0.83 HTR1A (0.43) HTR7ADRB1HTR3AHTR3EHTR3B
SCHEMBL9119904 0.83 HTR6 (0.46) HTR7ADRB1HTR1A
SCHEMBL1477092 0.74 ADRB1 (0.47) HTR7ADRB1
SCHEMBL2545151 0.72 HTR6 (0.47) HTR7ADRB1HTR1A
SCHEMBL31051724 0.69 DRD2 (0.67) HTR7ADRB1HTR3AHTR3EHTR3B
SCHEMBL22542051 0.68 ADRB1 (0.70) HTR7ADRB1HTR3AHTR3EHTR3B
SCHEMBL14904817 0.68 HTR7 (1.00) HTR7ADRB1HTR3AHTR1A
Hydrochloric Acid SCHEMBL27907732 0.67 ADRB1 (0.68) HTR7ADRB1HTR3AHTR3EHTR3B
SCHEMBL255197 0.67 HTR3A (0.67) HTR7ADRB1HTR3AHTR3EHTR3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0189612-B1 NEW PHARMACEUTICAL COMPOSITIONS HAVING A PSYCHOTROPIC ACTIVITY DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1992-11-04 EP claimed
EP-0189612-A1 New pharmaceutical compositions having a psychotropic activity DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1986-08-06 EP claimed
US-5424313-A Bibyclic heteroacrylpiperazine derivatives having psychotropic activity, and pharmaceutical compositions containing these derivatives DUPHAR INTERNATIONAL RESEARCH B.V. (NL) 1995-06-13 US disclosed
EP-0189612-B1 NEW PHARMACEUTICAL COMPOSITIONS HAVING A PSYCHOTROPIC ACTIVITY DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1992-11-04 EP disclosed
EP-0189612-A1 New pharmaceutical compositions having a psychotropic activity DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1986-08-06 EP disclosed