SCHEMBL9214875

SCHEMBL9214875

CC(C)(C)OC(=O)N[C@@H](CC(=O)OCc1ccccc1)C(=O)NCCc1ccc(C(=O)OCc2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CTSS P25774 5/20 0.51
CTSK P43235 4/20 0.51
CA2 P00918 3/20 0.51
KLK7 P49862 1/20 0.50
KLK5 Q9Y337 1/20 0.50
CA5A P35218 1/20 0.49
PPARA Q07869 2/20 0.48
PPARG P37231 1/20 0.48
CTSL P07711 1/20 0.48
CTSB P07858 1/20 0.48
AKT1 P31749 1/20 0.47
SYK P43405 1/20 0.47
CA1 P00915 1/20 0.47
PSMB1 P20618 1/20 0.45
PSMB8 P28062 1/20 0.45
PSMB9 P28065 1/20 0.45
PSMB5 P28074 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9224778 0.87 PSMB5 (0.51) CTSSCTSKCA2KLK7KLK5
SCHEMBL7404441 0.87 KLK7 (0.51) CTSSCTSKCA2KLK7KLK5
SCHEMBL15259723 0.85 MEN1 (0.56) CTSSCTSKKLK7KLK5CTSL
SCHEMBL9224769 0.85 KLK7 (0.45) CTSSCTSKCA2KLK7KLK5
SCHEMBL5656256 0.84 CTSK (0.54) CTSSCTSKCA2KLK7KLK5
SCHEMBL26294280 0.83 CA5A (0.55) CTSSCTSKCA2CA5ACTSL
SCHEMBL10825282 0.83 MEN1 (0.62) CTSSCTSKKLK7KLK5
Trifluoroacetic Acid SCHEMBL7703706 0.83 CA2 (0.49) CTSSCTSKCA2KLK7KLK5
SCHEMBL13108630 0.83 CTSS (0.57) CTSSCTSKKLK7KLK5PPARA
SCHEMBL9220637 0.83 CASP1 (0.55) CTSSCTSKCA2KLK7KLK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed