SCHEMBL9224778

SCHEMBL9224778

C[C@H](NC(=O)OC(C)(C)C)C(=O)N[C@@H](CC(=O)OCc1ccccc1)C(=O)NCCc1ccc(C(=O)O)cc1

nearest known ligand 0.51

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PSMB5 P28074 2/20 0.51
PSMB1 P20618 1/20 0.51
PSMB8 P28062 1/20 0.51
PSMB9 P28065 1/20 0.51
MMP8 P22894 1/20 0.47
CA2 P00918 4/20 0.46
CA5A P35218 2/20 0.46
CTSS P25774 4/20 0.46
CTSK P43235 3/20 0.46
PSMB10 P40306 1/20 0.46
PSMB2 P49721 1/20 0.46
KLK7 P49862 1/20 0.46
KLK5 Q9Y337 1/20 0.46
REN P00797 2/20 0.43
PPARG P37231 1/20 0.43
PPARA Q07869 1/20 0.43
CTSL P07711 1/20 0.43
CTSB P07858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9214875 0.87 CTSS (0.51) PSMB5PSMB1PSMB8PSMB9CA2
SCHEMBL9224769 0.87 KLK7 (0.45) PSMB5PSMB1PSMB8PSMB9MMP8
SCHEMBL7404441 0.82 KLK7 (0.51) PSMB5PSMB1PSMB8PSMB9CA2
SCHEMBL11648764 0.81 KLK5 (0.52) CTSSCTSKKLK7KLK5REN
SCHEMBL9220259 0.81 REN (0.55) CTSSCTSKKLK7KLK5REN
SCHEMBL28673197 0.80 KLK7 (0.53) MMP8CTSSCTSKKLK7KLK5
SCHEMBL28673199 0.80 KLK7 (0.53) MMP8CTSSCTSKKLK7KLK5
SCHEMBL26294280 0.79 CA5A (0.55) CA2CA5ACTSSCTSKCTSL
SCHEMBL15259723 0.78 MEN1 (0.56) CTSSCTSKKLK7KLK5CTSL
Trifluoroacetic Acid SCHEMBL7703706 0.78 CA2 (0.49) CA2CA5ACTSSCTSKKLK7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed