SCHEMBL9218199

SCHEMBL9218199

CC(C)(C)OC(=O)C[C@H](NC(=O)CCCc1ccc(C(=O)NS)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MMP1 P03956 1/20 0.49
MMP3 P08254 1/20 0.49
MMP9 P14780 1/20 0.49
KLK5 Q9Y337 1/20 0.44
MAPT P10636 2/20 0.42
TDP1 Q9NUW8 2/20 0.42
ACE P12821 1/20 0.42
POLB P06746 1/20 0.42
ROCK2 O75116 2/20 0.42
CTSG P08311 1/20 0.41
CMA1 P23946 1/20 0.41
HDAC1 Q13547 4/20 0.41
HDAC6 Q9UBN7 4/20 0.41
PSMB5 P28074 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7307254 0.88 MMP1 (0.49) MMP1MMP3MMP9KLK5MAPT
Iodide SCHEMBL9223621 0.80 MAPT (0.43) MMP1MMP3MMP9KLK5MAPT
Iodide SCHEMBL9223883 0.79 CCKBR (0.43) MMP1MMP3MMP9KLK5MAPT
SCHEMBL7302254 0.79 TDP1 (0.46) MMP1MMP3MMP9KLK5MAPT
SCHEMBL7296817 0.79 MAPT (0.44) MMP1MMP3MMP9KLK5MAPT
Iodide SCHEMBL9221941 0.78 CCKBR (0.43) MMP1MMP3MMP9KLK5MAPT
SCHEMBL9215215 0.78 ITGB3 (0.52) MMP1MMP3MMP9MAPTTDP1
SCHEMBL7301659 0.78 CTSG (0.46) MAPTTDP1CTSGCMA1PSMB5
SCHEMBL4941724 0.78 ACE (0.58) MMP1MMP3MMP9KLK5MAPT
Iodide SCHEMBL9215204 0.78 ITGB3 (0.51) MMP1MMP3MMP9MAPTTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed