SCHEMBL9268118

SCHEMBL9268118

COC1CCOC(c2cccc(COc3ccc4c(c3)OC(=O)CC4c3ccccc3)c2)C1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 9/20 0.48
ALDH2 P05091 1/20 0.46
MAPT P10636 4/20 0.43
MEN1 O00255 4/20 0.41
KMT2A Q03164 4/20 0.41
HPGD P15428 3/20 0.39
GAA P10253 1/20 0.39
HSD17B10 Q99714 1/20 0.39
THRB P10828 1/20 0.38
MAOB P27338 3/20 0.38
GRM5 P41594 2/20 0.38
NPC1 O15118 1/20 0.38
NFKB1 P19838 1/20 0.38
RAB9A P51151 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
HTR2B P41595 1/20 0.37
TMEM97 Q5BJF2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9259277 0.77 RAB9A (0.61) MEN1KMT2AMAOBNPC1RAB9A
SCHEMBL9158037 0.77 KMT2A (0.41) ALDH1A1MAPTKMT2AHPGDMAOB
SCHEMBL9263722 0.77 NPC1 (0.58) MEN1KMT2AMAOBNPC1RAB9A
SCHEMBL7662912 0.77 ALDH1A1 (0.64) ALDH1A1ALDH2MAPTMEN1KMT2A
SCHEMBL9254545 0.76 MAOB (0.61) ALDH1A1MEN1KMT2AHPGDMAOB
SCHEMBL9159704 0.76 KMT2A (0.41) MEN1KMT2AMAOBGRM5NPC1
SCHEMBL9156479 0.76 ALOX5 (0.38) ALDH1A1MEN1KMT2AHPGDMAOB
SCHEMBL9160911 0.76 MEN1 (0.44) MEN1KMT2AMAOBGRM5NPC1
SCHEMBL9161622 0.75 MAOB (0.39) ALDH1A1HPGDHSD17B10MAOBGRM5
SCHEMBL9159373 0.75 ALOX5 (0.49) MEN1KMT2AMAOBGRM5NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5424320-A Antihistamine, antiallergic, antiinflammatory and cytoprotective agents MERCK FROSST CANADA, INC. (CA) 1995-06-13 US claimed
US-5360815-A Heteroaryl cinnamic acids as inhibitors of leukotriene biosynthesis MERCK FROSST CANADA, INC. (CA) 1994-11-01 US disclosed