SCHEMBL9299028

SCHEMBL9299028

NC(=O)N(O)Cc1cccc(C(O)C#Cc2cccnc2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGES O14684 4/20 0.45
AKR1C3 P42330 2/20 0.43
FFAR1 O14842 1/20 0.38
CYP2A6 P11509 3/20 0.37
CYP2E1 P05181 2/20 0.36
CYP3A4 P08684 2/20 0.36
CYP2D6 P10635 2/20 0.36
CYP2C9 P11712 2/20 0.36
CYP2B6 P20813 2/20 0.36
CYP2C19 P33261 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C8 P10632 1/20 0.36
GRM2 Q14416 1/20 0.35
ALOX5 P09917 2/20 0.35
CHRNB2 P17787 2/20 0.34
CHRNA4 P43681 2/20 0.34
RECQL P46063 1/20 0.34
KDM4E B2RXH2 1/20 0.34
PKM P14618 1/20 0.34
PSMB5 P28074 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9299750 0.88 FFAR1 (0.43) PTGESAKR1C3FFAR1CYP2A6CYP2E1
SCHEMBL9299307 0.88 ALOX5 (0.41) PTGESALOX5
SCHEMBL9299828 0.81 ALOX5 (0.36) FFAR1ALOX5
SCHEMBL9300259 0.80 ACHE (0.39) PTGESALOX5KDM4E
SCHEMBL9300599 0.79 ALDH1A1 (0.43) PTGESAKR1C3FFAR1ALOX5PKM
SCHEMBL9299128 0.76 FFAR1 (0.43) PTGESAKR1C3FFAR1CYP2A6CYP2E1
SCHEMBL9300627 0.76 ALOX5 (0.45) PTGESALOX5
SCHEMBL8775926 0.74 NR3C2 (0.44) PTGESGRM2PSMB5
SCHEMBL9299972 0.74 ALOX5 (0.40) FFAR1ALOX5
SCHEMBL9299499 0.73 PTGES (0.42) PTGESCYP2C9ALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5326902-A Oxyalkyne compounds, pharmaceutical compositions containing them and processes for preparing such compounds and compositions GRUENENTHAL GMBH (DE) 1994-07-05 US disclosed