SCHEMBL9302190

SCHEMBL9302190

O=C(c1cccc(Cl)c1)N1CCC(CNCC2CSc3ccccc3O2)CC1

nearest known ligand 0.53

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MGLL Q99685 2/20 0.45
UBE2M P61081 1/20 0.44
DCUN1D1 Q96GG9 1/20 0.44
ADRB2 P07550 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C19 P33261 1/20 0.44
HSD11B1 P28845 1/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
ADRA1A P35348 2/20 0.42
ADRA1D P25100 1/20 0.42
ADRA1B P35368 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301424 0.90 ADRA1A (0.45) CYP2D6CYP2C19MEN1KMT2AADRA1A
SCHEMBL9302364 0.90 EPHX2 (0.46) MGLLUBE2MDCUN1D1CYP2D6CYP2C19
SCHEMBL9301904 0.87 ADRA1A (0.51) MGLLUBE2MDCUN1D1CYP2D6CYP2C19
SCHEMBL9302003 0.85 ADRA1D (0.60) MGLLADRA1AADRA1DADRA1B
SCHEMBL9302459 0.81 CXCR4 (0.54) CYP2D6CYP2C19ADRA1AADRA1DADRA1B
SCHEMBL9302183 0.77 CYP2D6 (0.44) MGLLUBE2MDCUN1D1ADRB2CYP2D6
SCHEMBL9301815 0.73 ADRA1D (0.63) ADRA1AADRA1DADRA1B
SCHEMBL9302076 0.73 EPHX2 (0.48) MGLLUBE2MDCUN1D1HSD11B1MEN1
SCHEMBL9302313 0.73 ADRA1D (0.57) ADRA1AADRA1DADRA1B
SCHEMBL9302494 0.73 ADRA1A (0.49) CYP2D6CYP2C19MEN1KMT2AADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5286735-A Antidepressants, anxiolytic agents PIERRE FABRE MEDICAMENT (FR) 1994-02-15 US claimed
US-5286735-A Antidepressants, anxiolytic agents PIERRE FABRE MEDICAMENT (FR) 1994-02-15 US disclosed