SCHEMBL9301180

SCHEMBL9301180

CN1CCN(c2c(F)c(NCc3ccccc3)c3c(c2F)n2c(=O)n(OCc4ccccc4)c(=O)cc2n3C2CC2)CC1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.36
IKBKB O14920 1/20 0.36
AURKA O14965 1/20 0.36
CHUK O15111 1/20 0.36
MAPK13 O15264 1/20 0.36
DAPK3 O43293 1/20 0.36
PRKCG P05129 1/20 0.36
PIM1 P11309 1/20 0.36
CDK2 P24941 1/20 0.36
MARK3 P27448 1/20 0.36
AKT1 P31749 1/20 0.36
AKT2 P31751 1/20 0.36
MAPKAPK2 P49137 1/20 0.36
GSK3A P49840 1/20 0.36
NEK2 P51955 1/20 0.36
PLK1 P53350 1/20 0.36
MAPK12 P53778 1/20 0.36
CDK5 Q00535 1/20 0.36
PRKCD Q05655 1/20 0.36
PAK1 Q13153 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301963 0.77 ALDH1A1 (0.36) HPGDMEN1USP2ALDH1A1LMNA
SCHEMBL9302110 0.69 ACHE (0.35) HTR6HRH4PDE5AHRH1HRH2
SCHEMBL9302877 0.68 GRM5 (0.39) HPGDSMN1; SMN2ALDH1A1LMNAKMT2A
SCHEMBL9302233 0.67 ALDH1A1 (0.39) HTR6HPGDMEN1USP2ALDH1A1
SCHEMBL9303411 0.67 ALDH1A1 (0.41) HPGDMEN1ALDH1A1LMNAKMT2A
SCHEMBL9302194 0.67 ACHE (0.39) HTR6IKBKBAURKACHUKMAPK13
SCHEMBL9302209 0.66 PIK3CD (0.35) HPGDSMN1; SMN2HRH3MEN1USP2
SCHEMBL29634202 0.64 TSHR (0.33) USP2ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL6796311 0.64 ALDH1A1 (0.41) HRH4MEN1USP2ALDH1A1LMNA
SCHEMBL9302522 0.63 SIRT6 (0.47) HTR6HRH4PDE5ANOD2NOD1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed