SCHEMBL9302144

SCHEMBL9302144

CN1CCN(c2cc3c(cc2F)nc(CC(=O)NOCc2ccccc2)n3C2CC2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.39
ALDH1A1 P00352 5/20 0.38
KDM4E B2RXH2 3/20 0.38
HPGD P15428 1/20 0.38
OPRM1 P35372 1/20 0.38
OPRD1 P41143 1/20 0.38
OPRK1 P41145 1/20 0.38
OGFRL1 Q5TC84 1/20 0.38
CPT1A P50416 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
CSF1R P07333 2/20 0.37
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
LMNA P02545 2/20 0.37
CYP11B1 P15538 1/20 0.37
CYP11B2 P19099 1/20 0.37
BRD4 O60885 1/20 0.36
CREBBP Q92793 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301969 0.92 GRM5 (0.42) GRM5ALDH1A1HPGDOPRM1OPRD1
SCHEMBL9302252 0.89 ACHE (0.42) GRM5OPRM1OPRD1OGFRL1LMNA
SCHEMBL9303370 0.87 ALDH1A1 (0.43) GRM5ALDH1A1KDM4EHPGDNPC1
SCHEMBL9303690 0.83 OPRM1 (0.37) OPRM1OPRD1OPRK1OGFRL1CPT1A
SCHEMBL9302311 0.81 CYP11B2 (0.44) ALDH1A1KDM4EHPGDNPC1CSF1R
Hydrochloric Acid SCHEMBL9302957 0.81 CYP11B1 (0.43) ALDH1A1KDM4EHPGDNPC1CSF1R
SCHEMBL9301930 0.79 HTT (0.45) ALDH1A1KDM4EHPGDSMN1; SMN2MEN1
Acetic Acid SCHEMBL9301936 0.78 CYP11B2 (0.44) ALDH1A1KDM4EHPGDNPC1MEN1
SCHEMBL9301682 0.75 RORC (0.42) OPRM1OPRD1OGFRL1SMN1; SMN2LMNA
SCHEMBL9303809 0.74 HTT (0.41) ALDH1A1OPRM1OPRD1OGFRL1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed