SCHEMBL9302110

SCHEMBL9302110

CN1CCN(c2c(F)c(NCc3ccccc3)c3c(nc(CC(=O)NOCc4ccccc4)n3C3CC3)c2F)CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.35
HTR6 P50406 3/20 0.35
HRH4 Q9H3N8 7/20 0.35
PDE5A O76074 1/20 0.35
HRH1 P35367 2/20 0.34
CTNNB1 P35222 1/20 0.34
TCF7L2 Q9NQB0 1/20 0.34
STAT6 P42226 1/20 0.33
JAK2 O60674 1/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
JAK3 P52333 1/20 0.33
BRD4 O60885 1/20 0.33
CREBBP Q92793 1/20 0.33
OPRM1 P35372 1/20 0.33
OPRD1 P41143 1/20 0.33
OPRK1 P41145 1/20 0.33
OGFRL1 Q5TC84 1/20 0.33
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302194 0.83 ACHE (0.39) ACHEHTR6HRH4PDE5AHRH1
SCHEMBL9302144 0.74 GRM5 (0.39) HRH4BRD4CREBBPOPRM1OPRD1
SCHEMBL9301180 0.69 HTR6 (0.36) ACHEHTR6HRH4PDE5AHRH1
SCHEMBL9301969 0.66 GRM5 (0.42) OPRM1OPRD1OPRK1OGFRL1
SCHEMBL9302252 0.65 ACHE (0.42) ACHEOPRM1OPRD1OGFRL1
SCHEMBL9303370 0.64 ALDH1A1 (0.43) HRH4
SCHEMBL9302522 0.62 SIRT6 (0.47) ACHEHTR6HRH4PDE5AJAK2
SCHEMBL7424713 0.58 NPC1 (0.62) EGFR
SCHEMBL7970712 0.56 NPC1 (0.62) EGFR
SCHEMBL906398 0.56 RAB9A (0.62) EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed