SCHEMBL9358666

SCHEMBL9358666

C#CC(I)OC(=O)CCC(=O)[O-].[Na+]

nearest known ligand 0.35

Known targets — ChEMBL curated mechanism

ABCC8ACEADORA1ADORA2AADORA2BADORA3ALDH5A1ALOX5ALOX5APATP4AATP4BBRAFCA1CA12CA2CA4CYSLTR1DHFRDPEP1EDNRAEDNRBESR2F10FDPSFGF1GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGARTGNRHRGSC1HMGCRIMPDH1IMPDH2KCNJ11LY96NOD2NR3C1NS3NS4ANS5bP2RY1P2RY12P2RY2P2RY4P2RY6PBP2XPDE3APDE3BPDE4APDE4BPDE4CPDE4DPDK1PDK2PDK3PDK4PPARGPPATPTGIRPTGS1PTGS2RAF1RYR1RYR3SCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASERPINC1SLC12A1SLC12A3SYKTHRATHRBTLR3TLR4TLR9TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYMSVKORC1XDHblablaIMP-1blaOXA-33blaOXA-58blaT-3blaT-4blaT-5blaT-6dacAdacBdacCfolAfolPfolP1ftsIfusAgaggyrAgyrBmecAmrcAmrcBmrdApbp1apbp1bpbp2pbp2apbp2bpbp3pbp4pbpApbpBpbpCpbpFpolponBrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpoArpoBrpoCrpoZrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CA1 known ✓ P00915 1/20 0.32
ELANE P08246 1/20 0.35
FFAR3 O14843 1/20 0.31
HDAC3 O15379 1/20 0.31
HDAC1 Q13547 1/20 0.31
HDAC2 Q92769 1/20 0.31
HDAC8 Q9BY41 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9621020 0.88 CYP2D6 (0.31)
SCHEMBL27514652 0.68 HDAC3 (0.43) ELANECA1FFAR3HDAC3HDAC1
SCHEMBL2353376 0.65 CA1 (0.43) ELANECA1FFAR3HDAC3HDAC1
SCHEMBL27801920 0.65 HDAC3 (0.46) ELANECA1FFAR3HDAC3HDAC1
Succinic Acid SCHEMBL24440 0.64 HDAC3 (0.62) CA1FFAR3HDAC3HDAC1HDAC2
Succinic Acid SCHEMBL3012461 0.64 HDAC3 (0.62) CA1FFAR3HDAC3HDAC1HDAC2
SCHEMBL30622578 0.62 FFAR3 (0.42) ELANECA1FFAR3HDAC3HDAC1
SCHEMBL16722616 0.62 FFAR3 (0.42) ELANECA1FFAR3HDAC3HDAC1
SCHEMBL15776451 0.62 HDAC3 (0.42) ELANECA1FFAR3HDAC3HDAC1
Succinic Acid SCHEMBL6249858 0.62 TSHR (0.68) CA1FFAR3HDAC3HDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0359442-B1 Mono-iodopropargyl esters of dicarboxylic anhydrides and their use as antimicrobial agents LONZA AG (US) 1994-10-19 EP disclosed
US-5073570-A MONO-IODOPROPARGYL ESTERS OF DICARBOXYLIC ANHYDRIDES AND THEIR USE AS ANTIMICROBIAL AGENTS LONZA INC. (US) 1991-12-17 US disclosed
EP-0359442-A2 Mono-iodopropargyl esters of dicarboxylic anhydrides and their use as antimicrobial agents LONZA INC. (US) 1990-03-21 EP disclosed