SCHEMBL9401169

SCHEMBL9401169

CCN(C(C)=O)c1c(Cc2ccccc2)[nH]c2ccc(OC)cc12

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTNR1A P48039 5/20 0.58
MTNR1B P49286 5/20 0.58
KMT2A Q03164 4/20 0.47
MEN1 O00255 2/20 0.47
ALDH1A1 P00352 5/20 0.44
KDM4E B2RXH2 4/20 0.44
POLB P06746 1/20 0.44
GAA P10253 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
FPR1 P21462 1/20 0.43
CYP1A2 P05177 2/20 0.42
CYP3A4 P08684 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
CYP2C19 P33261 2/20 0.42
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42
AHR P35869 1/20 0.42
AKR1C2 P52895 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9401142 0.87 KMT2A (0.49) MTNR1AMTNR1BKMT2AMEN1ALDH1A1
SCHEMBL9401130 0.84 MTNR1A (0.51) MTNR1AMTNR1BKMT2AMEN1ALDH1A1
SCHEMBL10444002 0.75 MTNR1A (0.67) MTNR1AMTNR1BKMT2AMEN1ALDH1A1
SCHEMBL9401166 0.74 MTNR1A (0.58) MTNR1AMTNR1BKMT2AMEN1ALDH1A1
SCHEMBL9304037 0.73 MTNR1A (1.00) MTNR1AMTNR1BKMT2AMEN1ALDH1A1
SCHEMBL8802574 0.70 MTNR1A (0.67) MTNR1AMTNR1BKMT2AMEN1ALDH1A1
SCHEMBL9535590 0.69 KDM4E (0.58) KMT2AMEN1ALDH1A1KDM4EPOLB
SCHEMBL8805501 0.68 MTNR1A (0.60) MTNR1AMTNR1BKMT2AMEN1ALDH1A1
SCHEMBL7696761 0.67 AKR1C2 (0.61) MTNR1AMTNR1BKMT2AMEN1ALDH1A1
SCHEMBL9145256 0.66 ALDH1A1 (0.53) KMT2AMEN1ALDH1A1KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5314908-A Compounds useful as antiproliferative agents WHITBY RESEARCH, INC. (US) 1994-05-24 US disclosed
EP-0549916-A2 Compounds useful as antiproliferative agents WHITBY RESEARCH, Inc. (US) 1993-07-07 EP disclosed
US-5206377-A Compounds useful as antiproliferative agents WHITBY RESEARCH, INC. (US) 1993-04-27 US disclosed