SCHEMBL9429583

SCHEMBL9429583

Cn1c(N2CCN(CCCOc3c(Cl)cc(C#N)cc3Cl)CC2)cc(=O)n(C)c1=O

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
KMT2A Q03164 1/20 0.44
HRH3 Q9Y5N1 7/20 0.40
HRH1 P35367 10/20 0.40
HRH2 P25021 4/20 0.39
KCNJ5 P48544 1/20 0.38
KCNJ3 P48549 1/20 0.38
CCR3 P51677 1/20 0.38
ADRA1A P35348 3/20 0.38
HTR1A P08908 2/20 0.38
DRD2 P14416 1/20 0.38
HTR2A P28223 1/20 0.38
HTR7 P34969 1/20 0.38
ADRA1D P25100 2/20 0.37
ADRA1B P35368 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9428870 0.85 HRH3 (0.57) MEN1ALDH1A1KMT2AHRH3HRH1
SCHEMBL9429616 0.82 HRH3 (0.58) MEN1ALDH1A1KMT2AHRH3HRH1
SCHEMBL9428883 0.82 HRH1 (0.50) MEN1ALDH1A1KMT2AHRH3HRH1
SCHEMBL9386451 0.82 ALDH1A1 (0.43) MEN1ALDH1A1KMT2AHRH3HRH1
Hydrochloric Acid SCHEMBL9386358 0.81 ALDH1A1 (0.42) MEN1ALDH1A1KMT2AHRH3HRH1
SCHEMBL9429324 0.81 DRD2 (0.56) HRH3HRH1HRH2HTR1ADRD2
Hydrochloric Acid SCHEMBL9428228 0.80 SIGMAR1 (0.55) HRH3HRH1HRH2HTR1ADRD2
SCHEMBL9428720 0.79 MEN1 (0.50) MEN1ALDH1A1KMT2AHRH3HRH1
SCHEMBL9428375 0.79 ALDH1A1 (0.43) MEN1ALDH1A1KMT2AADRA1AHTR1A
SCHEMBL9428864 0.79 KDM4E (0.57) MEN1ALDH1A1KMT2AHRH1ADRA1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5332739-A Pyrimidinedione derivatives and antiarrhythmic agents containing same MITSUI TOATSU CHEMICALS, INCORPORATED (JP) 1994-07-26 US disclosed