SCHEMBL9448992

SCHEMBL9448992

[N-]=[N+]=CC(=O)c1ccccc1-c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.52
GPR52 Q9Y2T5 1/20 0.49
MEN1 O00255 3/20 0.47
KMT2A Q03164 3/20 0.47
SMN1; SMN2 Q16637 2/20 0.47
CHRNB2 P17787 3/20 0.46
CHRNB4 P30926 3/20 0.46
CHRNA3 P32297 3/20 0.46
CHRNA4 P43681 3/20 0.46
HNF4A P41235 1/20 0.44
TSHR P16473 1/20 0.44
RECQL P46063 1/20 0.44
NPSR1 Q6W5P4 2/20 0.43
HSP90AA1 P07900 1/20 0.42
FABP3 P05413 1/20 0.41
FABP4 P15090 1/20 0.41
FABP5 Q01469 1/20 0.41
ALDH1A1 P00352 4/20 0.41
HTT P42858 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6169408 0.80 SLC22A12 (0.43) HTT
SCHEMBL7613879 0.79 ALDH1A1 (0.56) MEN1KMT2ASMN1; SMN2NPSR1ALDH1A1
SCHEMBL7864455 0.77 BCAT2 (0.59) BCAT2GPR52MEN1KMT2ASMN1; SMN2
SCHEMBL5180034 0.76 BCAT2 (0.57) BCAT2GPR52MEN1KMT2ASMN1; SMN2
SCHEMBL31521259 0.76 BCAT2 (0.57) BCAT2GPR52MEN1KMT2ASMN1; SMN2
SCHEMBL9448980 0.74 CES2 (0.52) GPR52MEN1KMT2ATSHRNPSR1
SCHEMBL9449288 0.74 CES2 (0.52) MEN1KMT2ATSHRRECQLNPSR1
SCHEMBL9448951 0.74 ALDH1A1 (0.46) MEN1KMT2ANPSR1HSP90AA1ALDH1A1
SCHEMBL9448877 0.74 GPR52 (0.45) GPR52MEN1KMT2ASMN1; SMN2NPSR1
SCHEMBL28340415 0.74 GPR52 (0.59) BCAT2GPR52MEN1KMT2ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0466730-B1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1993-07-21 EP disclosed
US-5220021-A Geminal bisphosphonic acids and derivatives as anti-arthritic agents THE UPJOHN COMPANY (US) 1993-06-15 US disclosed
WO-1990012017-A1 GEMINAL BISPHOSPHONIC ACIDS AND DERIVATIVES AS ANTI-ARTHRITIC AGENTS THE UPJOHN COMPANY (US) 1990-10-18 WO disclosed