SCHEMBL9490432

SCHEMBL9490432

O=C(O)CN1C(=O)CN(S(=O)(=O)c2ccc(F)cc2)c2ccccc21

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP2 P08253 2/20 0.54
ALDH1A1 P00352 6/20 0.49
MEN1 O00255 3/20 0.49
KMT2A Q03164 3/20 0.49
GAA P10253 3/20 0.49
HPGD P15428 2/20 0.49
MCOLN3 Q8TDD5 1/20 0.49
CTSG P08311 1/20 0.44
CMA1 P23946 1/20 0.44
PKM P14618 3/20 0.43
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
CHRNB2 P17787 1/20 0.41
CHRNB4 P30926 1/20 0.41
CHRNA3 P32297 1/20 0.41
CHRNA4 P43681 1/20 0.41
MAPT P10636 2/20 0.40
POLB P06746 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9490572 0.91 MMP2 (0.55) MMP2ALDH1A1MEN1KMT2APKM
SCHEMBL9490689 0.88 MMP2 (0.54) MMP2ALDH1A1MEN1KMT2ACTSG
SCHEMBL9490445 0.88 MMP2 (0.54) MMP2ALDH1A1MEN1KMT2AGAA
SCHEMBL9489398 0.85 MMP2 (0.56) MMP2ALDH1A1CTSGCMA1PKM
SCHEMBL9699725 0.84 NPSR1 (0.49) MMP2ALDH1A1MEN1KMT2AGAA
SCHEMBL9490595 0.78 CTSG (0.44) MMP2ALDH1A1MEN1KMT2ACTSG
SCHEMBL9490990 0.76 NPSR1 (0.53) MMP2ALDH1A1MEN1KMT2AGAA
Acetic Acid SCHEMBL10461101 0.76 MMP2 (0.53) MMP2ALDH1A1MEN1KMT2AGAA
SCHEMBL10459002 0.74 L3MBTL1 (0.50) ALDH1A1MEN1KMT2AGAAPKM
SCHEMBL9697221 0.74 KMT2A (0.53) MMP2ALDH1A1MEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0266102-B1 QUINOXALINONE DERIVATIVES PFIZER INC. (US) 1993-03-17 EP disclosed
US-4940708-A 4-arylsulfonyl-3,4-dihydro-2(1H)-quinoxalinone-1-alkanoic acids, esters, and salts PFIZER INC. (US) 1990-07-10 US disclosed