SCHEMBL9701972

SCHEMBL9701972

CC1=Nc2c(N(C)Cc3ccc(S(=O)(=O)c4ccccc4)cc3)ccc3cccc(c23)N1

nearest known ligand 0.53

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TYMS P04818 9/20 0.53
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
MCL1 Q07820 1/20 0.39
SCN9A Q15858 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HTR6 P50406 1/20 0.32
FFAR2 O15552 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9508035 0.71 TYMS (0.55) TYMSSCN9AHTR6FFAR2
SCHEMBL16506969 0.66 GAA (0.62) GAAMAPTMCL1ALDH1A1
SCHEMBL12083406 0.64 ALDH1A1 (0.59) TYMSGAAMAPTALDH1A1HTR6
SCHEMBL4664193 0.63 TYMS (0.46) TYMSGAAMAPTALDH1A1HTR6
SCHEMBL9508011 0.63 TYMS (0.73) TYMSSCN9A
SCHEMBL9508662 0.63 TYMS (0.59) TYMSMAPTALDH1A1
SCHEMBL9080571 0.61 TYMS (0.79) TYMSMAPTALDH1A1
SCHEMBL4664189 0.61 TYMS (0.46) TYMSGAAMAPTALDH1A1HTR6
SCHEMBL9504568 0.60 TYMS (0.69) TYMSALDH1A1HTR6FFAR2
SCHEMBL9587910 0.59 DHFR (0.47) TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992005153-A1 ANTIPROLIFERATIVE SUBSTITUTED NAPHTHALENE COMPOUNDS AGOURON PHARMACEUTICALS, INC. (US) 1992-04-02 WO disclosed