SCHEMBL9533388

SCHEMBL9533388

Cc1cccc(NC(=O)Oc2c(-c3ccccc3)noc2C)c1C

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 5/20 0.51
HTT P42858 1/20 0.51
NPC1 O15118 4/20 0.47
RAB9A P51151 3/20 0.47
MAPT P10636 3/20 0.45
RXFP1 Q9HBX9 2/20 0.44
ALDH1A1 P00352 4/20 0.44
NPSR1 Q6W5P4 2/20 0.43
KDM4E B2RXH2 1/20 0.43
HPGD P15428 1/20 0.43
CASP1 P29466 1/20 0.43
CASP7 P55210 1/20 0.43
UBE2N P61088 1/20 0.43
HSD17B10 Q99714 1/20 0.43
LMNA P02545 1/20 0.43
GAA P10253 2/20 0.43
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2C19 P33261 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9534238 0.83 POLB (0.45) TSHRHTTMAPTNPSR1KDM4E
SCHEMBL9535755 0.80 ALDH1A1 (0.52) MAPTALDH1A1GAACYP1A2CYP2C19
SCHEMBL9533884 0.79 KMT2A (0.59) TSHRHTTNPC1MAPTRXFP1
SCHEMBL9533937 0.78 ALDH1A1 (0.50) HTTMAPTALDH1A1KDM4EKMT2A
SCHEMBL9536170 0.78 MAPT (0.52) TSHRMAPTALDH1A1KDM4EKMT2A
SCHEMBL9537484 0.77 LMNA (0.52) TSHRHTTMAPTALDH1A1NPSR1
SCHEMBL5242546 0.77 KMT2A (0.56) TSHRHTTGAAKMT2AMEN1
SCHEMBL27495331 0.76 KMT2A (0.55) TSHRHTTALDH1A1GAAKMT2A
SCHEMBL9533918 0.75 MAPT (0.64) HTTNPC1RAB9AMAPTALDH1A1
SCHEMBL9535701 0.74 KMT2A (0.54) TSHRHTTGAAKMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0573883-A1 Utilization of 3 substituted aryl-5-alkyl-isoxazole-4-carboxylic acid derivatives against endoparasites new 3-substituted aryl-5-alkyl-isoxazole-4-carboxylic acid derivatives and process for their preparation BAYER AG (DE) 1993-12-15 EP disclosed