SCHEMBL9537454

SCHEMBL9537454

Cc1ccc(NC(=O)Oc2c(-c3ccc(Cl)cc3)noc2C)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 1/20 0.50
GPBAR1 Q8TDU6 3/20 0.49
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
NPC1 O15118 2/20 0.43
ALDH1A1 P00352 2/20 0.43
CYP3A4 P08684 2/20 0.43
AURKA O14965 1/20 0.43
RAB9A P51151 4/20 0.43
CNR1 P21554 1/20 0.42
PTGS2 P35354 1/20 0.42
ATM Q13315 1/20 0.42
TRPV1 Q8NER1 1/20 0.42
CYP1A2 P05177 1/20 0.42
GAA P10253 1/20 0.42
CYP2C9 P11712 1/20 0.42
ALOX12 P18054 1/20 0.42
CYP2C19 P33261 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
POLB P06746 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9536170 0.91 MAPT (0.52) GHSRGPBAR1MEN1KMT2AALDH1A1
SCHEMBL9535755 0.88 ALDH1A1 (0.52) GHSRALDH1A1CYP3A4PTGS2CYP1A2
SCHEMBL9537105 0.85 MAPT (0.56) GPBAR1MEN1KMT2ANPC1ALDH1A1
SCHEMBL9534238 0.81 POLB (0.45) GHSRGPBAR1MEN1KMT2ACYP3A4
SCHEMBL9533383 0.79 GPBAR1 (0.51) GHSRGPBAR1MEN1KMT2ANPC1
SCHEMBL9533937 0.79 ALDH1A1 (0.50) GHSRMEN1KMT2AALDH1A1SMN1; SMN2
SCHEMBL9533918 0.76 MAPT (0.64) MEN1KMT2ANPC1ALDH1A1CYP3A4
SCHEMBL10192035 0.73 KMT2A (0.55) MEN1KMT2ANPC1ALDH1A1CYP3A4
SCHEMBL9535442 0.71 GPBAR1 (0.51) GPBAR1MEN1KMT2ANPC1ALDH1A1
SCHEMBL9533943 0.70 GHSR (0.54) GHSRPTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0573883-A1 Utilization of 3 substituted aryl-5-alkyl-isoxazole-4-carboxylic acid derivatives against endoparasites new 3-substituted aryl-5-alkyl-isoxazole-4-carboxylic acid derivatives and process for their preparation BAYER AG (DE) 1993-12-15 EP disclosed