SCHEMBL9537893

SCHEMBL9537893

COc1cc(N)c(N)c(Cc2ccco2)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.41
HPGD P15428 4/20 0.41
HSD17B10 Q99714 2/20 0.41
KDM4E B2RXH2 1/20 0.41
TSHR P16473 1/20 0.40
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
GAA P10253 2/20 0.39
ALOX12 P18054 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP19A1 P11511 1/20 0.38
POLB P06746 3/20 0.38
LMNA P02545 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.37
TAS1R3 Q7RTX0 1/20 0.36
TAS1R1 Q7RTX1 1/20 0.36
MAPT P10636 1/20 0.36
ALOX15 P16050 1/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9536206 0.74 TXNRD1 (0.37) ALDH1A1HPGDHSD17B10KDM4EMEN1
SCHEMBL24172156 0.71 ALDH1A1 (0.44) ALDH1A1HPGDHSD17B10KDM4ETSHR
SCHEMBL9539903 0.70 L3MBTL1 (0.42) ALDH1A1MEN1KMT2AL3MBTL1SMN1; SMN2
SCHEMBL28091649 0.69 LTA4H (0.55) ALDH1A1HPGDHSD17B10KDM4ETSHR
SCHEMBL9536141 0.69 LMNA (0.39) ALDH1A1HPGDHSD17B10KDM4EMEN1
SCHEMBL6912345 0.69 GAA (0.41) ALDH1A1HPGDKDM4ETSHRMEN1
SCHEMBL11035894 0.69 LMNA (0.54) ALDH1A1HPGDHSD17B10KDM4ETSHR
SCHEMBL21401837 0.68 CHRM2 (0.49) ALDH1A1HPGDHSD17B10TSHRMEN1
SCHEMBL2875800 0.68 GAA (0.45) ALDH1A1HPGDKDM4ETSHRMEN1
SCHEMBL25082470 0.67 GPR84 (0.69) KDM4ETSHRL3MBTL1MAPTNPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0151826-B1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1993-03-31 EP disclosed
EP-0151826-A1 4-[(Bicyclic heterocyclyl)-methyl and -hetero]-piperidines JANSSEN PHARMACEUTICA N.V. (BE) 1985-08-21 EP disclosed