SCHEMBL9541398

SCHEMBL9541398

CC=Cn1c(Cc2ccc(Br)cc2)c(CC)c2c(O)cccc2c1=O

nearest known ligand 0.34

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
VKORC1 Q9BQB6 1/20 0.34
PDE3B Q13370 2/20 0.31
PDE3A Q14432 2/20 0.31
ALOX5 P09917 1/20 0.31
PARP1 P09874 1/20 0.30
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9541340 0.73 PDE3B (0.37) VKORC1PDE3BPDE3A
SCHEMBL9542605 0.71 ALOX5 (0.42) VKORC1PDE3BPDE3AALOX5PARP1
SCHEMBL9539844 0.67 PDE3B (0.37) VKORC1PDE3BPDE3A
SCHEMBL9542481 0.56 HSD17B10 (0.37)
SCHEMBL12834567 0.55 STAT3 (0.49) MAOB
SCHEMBL27561174 0.55 ALDH1A1 (0.40)
SCHEMBL4814389 0.55 TRPA1 (0.45)
SCHEMBL7205047 0.54 MAPT (0.46) PARP1
SCHEMBL2250646 0.54 KEAP1 (0.70) ALOX5
SCHEMBL68691 0.53 GABRA1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1993014086-A1 SUBSTITUTED 1-ISOQUINOLONE DERIVATIVES AS ANGIOTENSIN II ANTAGONISTS SYNTEX (U.S.A.) INC. (US) 1993-07-22 WO disclosed