SCHEMBL9541963

SCHEMBL9541963

COc1ccc(C=P(c2ccccc2)(c2ccccc2)c2ccccc2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.57
CA4 P22748 1/20 0.48
LTA4H P09960 2/20 0.47
ALDH1A1 P00352 2/20 0.45
CYP2A6 P11509 1/20 0.45
G6PC1 P35575 1/20 0.45
CYP3A4 P08684 2/20 0.44
LMNA P02545 1/20 0.44
TP53 P04637 1/20 0.44
TSHR P16473 1/20 0.44
KDM4E B2RXH2 1/20 0.44
RELA Q04206 5/20 0.44
BCHE P06276 1/20 0.44
NFKB1 P19838 1/20 0.44
NFKB2 Q00653 1/20 0.44
SERPINE1 P05121 1/20 0.44
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14423637 0.82 LTA4H (0.48) LTA4HALDH1A1LMNATSHRCA1
SCHEMBL1132385 0.79 ALDH1A1 (0.39) TRPA1CA4ALDH1A1CYP2A6LMNA
SCHEMBL9538596 0.78 LMNA (0.42) ALDH1A1CYP2A6CYP3A4LMNATSHR
SCHEMBL9539397 0.75 ALDH1A1 (0.41) ALDH1A1CYP3A4LMNATP53CA1
SCHEMBL11707690 0.74 TSHR (0.56) ALDH1A1LMNATSHRCA12CA1
SCHEMBL24193844 0.74 ESR1 (0.50) CA4ALDH1A1G6PC1CYP3A4RELA
SCHEMBL14269409 0.74 ALDH1A1 (0.42) TRPA1ALDH1A1CYP2A6LMNACYP1B1
SCHEMBL9541503 0.74 TSHR (0.42) CYP2A6G6PC1LMNATSHRNFE2L2
SCHEMBL9541494 0.74 NFE2L2 (0.52) ALDH1A1TSHRRELANFKB1NFKB2
SCHEMBL9538770 0.73 TRPV1 (0.41) LMNATSHRCA1CA2CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1104405-B1 NEAR INFRARED CHEMILUMINESCENT ACRIDINIUM COMPOUNDS AND USES THEREOF SIEMENS HEALTHCARE DIAGNOSTICS (US) 2009-02-18 EP disclosed
EP-0311955-B1 BICYCLIC PEROXIDE F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
US-5134240-A Malaria therapy HOFFMANN-LAROCHE, INC. (US) 1992-07-28 US disclosed
US-4977184-A Bicyclic peroxides compositions for and treatment of malaria therewith HOFFMANN-LA ROCHE INC. (US) 1990-12-11 US disclosed
EP-0311955-A2 Bicyclic peroxide F. HOFFMANN-LA ROCHE AG (CH) 1989-04-19 EP disclosed
US-4065620-A ANTIBIOTICS ELI LILLY AND COMPANY (US) 1977-12-27 US disclosed