SCHEMBL9588274

SCHEMBL9588274

CC1(C)C=Cc2cc(C(F)(F)F)ccc2C1=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 3/20 0.39
AR P10275 1/20 0.35
ABCC9 O60706 1/20 0.33
ABCC8 Q09428 1/20 0.33
KCNJ11 Q14654 1/20 0.33
KCNJ8 Q15842 1/20 0.33
MAPT P10636 2/20 0.33
PARP1 P09874 1/20 0.33
PARP10 Q53GL7 1/20 0.33
GPR3 P46089 1/20 0.33
NOTUM Q6P988 1/20 0.32
HSD17B10 Q99714 1/20 0.31
CES2 O00748 2/20 0.31
KDM4E B2RXH2 2/20 0.31
APAF1 O14727 1/20 0.31
NSD2 O96028 1/20 0.31
CASP3 P42574 1/20 0.31
GALK1 P51570 1/20 0.31
BLM P54132 1/20 0.31
KMT2A Q03164 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9587759 0.88 ABCC9 (0.44) ABCC9ABCC8KCNJ11KCNJ8
SCHEMBL9587106 0.75 PPOX (0.40) CYP11B2
SCHEMBL9588381 0.75 CA2 (0.42) TDP2PARP10
SCHEMBL30828314 0.72 TDP2 (0.41) TDP2MAPTPARP1PARP10GPR3
SCHEMBL4228062 0.70 ALDH1A1 (0.42) TDP2MAPTHSD17B10CES2KDM4E
SCHEMBL9731044 0.68 PDE2A (0.34) ARMAPTHSD17B10CES2KDM4E
SCHEMBL10838748 0.66 PGR (0.47) TDP2ARMAPTHSD17B10KMT2A
SCHEMBL7766906 0.66 ALDH1A1 (0.42) MAPTHSD17B10KDM4E
SCHEMBL12261410 0.66 TDP2 (0.50) TDP2PARP1PARP10NOTUMCYP11B2
SCHEMBL9565010 0.65 CA1 (0.42) KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5272170-A Tetralones with pharmacological activity J. URIACH & CIA., S.A. (ES) 1993-12-21 US disclosed
US-5208246-A Hypotensive, bronchodilator J. URIACH & CIA. (ES) 1993-05-04 US disclosed
EP-0489300-A2 Tetralones with pharmacological activity J. URIACH & CIA. S.A. (ES) 1992-06-10 EP disclosed