SCHEMBL9609465

SCHEMBL9609465

N[C@@H](Cc1c[nH]c2ccccc12)C(=O)Nc1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.71
KMT2A Q03164 3/20 0.71
MAPT P10636 3/20 0.71
KDM4E B2RXH2 2/20 0.71
LMNA P02545 1/20 0.71
MPO P05164 1/20 0.71
TSHR P16473 1/20 0.71
BLM P54132 1/20 0.71
PMP22 Q01453 1/20 0.71
HIF1A Q16665 1/20 0.71
RUVBL1 Q9Y265 4/20 0.68
AKT1 P31749 2/20 0.61
CDC7 O00311 1/20 0.61
CHUK O15111 1/20 0.61
MAPK13 O15264 1/20 0.61
DAPK3 O43293 1/20 0.61
DYRK3 O43781 1/20 0.61
ROCK2 O75116 1/20 0.61
RPS6KA5 O75582 1/20 0.61
PRKCG P05129 1/20 0.61

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9610738 1.00 MEN1 (0.71) MEN1KMT2AMAPTKDM4ELMNA
SCHEMBL30767397 1.00 MEN1 (0.71) MEN1KMT2AMAPTKDM4ELMNA
Hydrochloric Acid SCHEMBL19747056 0.99 MEN1 (0.69) MEN1KMT2AMAPTKDM4ELMNA
Hydrochloric Acid SCHEMBL21082966 0.99 MEN1 (0.69) MEN1KMT2AMAPTKDM4ELMNA
Hydrochloric Acid SCHEMBL19748758 0.95 RUVBL1 (0.73) MEN1KMT2AMAPTKDM4ELMNA
SCHEMBL11860142 0.92 RUVBL1 (0.65) MEN1KMT2AMAPTKDM4ELMNA
SCHEMBL28072305 0.92 RUVBL1 (0.65) MEN1KMT2AMAPTKDM4ELMNA
SCHEMBL8252240 0.91 RUVBL1 (0.70) MEN1KMT2AMAPTKDM4ELMNA
Hydrochloric Acid SCHEMBL19748580 0.91 RUVBL1 (0.63) MEN1KMT2AMAPTKDM4ELMNA
Hydrochloric Acid SCHEMBL19748954 0.91 RUVBL1 (0.63) MEN1KMT2AMAPTKDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117603084-A Peptidase neurolysin enhancer and preparation method and application thereof 江苏瑞思坦生物科技有限公司 2024-02-27 CN claimed
CN-117603084-A Peptidase neurolysin enhancer and preparation method and application thereof 江苏瑞思坦生物科技有限公司 2024-02-27 CN disclosed
US-8674144-B2 Catalyst for asymmetric hydrogenation and method for manufacturing optically active carbonyl compound using the same TAKASAGO INTERNATIONAL CORPORATION (JP) 2014-03-18 US disclosed
US-8674144-B2 Catalyst for asymmetric hydrogenation and method for manufacturing optically active carbonyl compound using the same TAKASAGO INTERNATIONAL CORPORATION (JP) 2014-03-18 US disclosed
EP-1865950-B1 COMPOUNDS USEFUL AS MODULATORS OF THE PROTEASOME ACTIVITY CENTRE NAT RECH SCIENT (FR) 2013-08-28 EP disclosed
US-20130196050-A1 SALTY TASTE ENHANCER AJINOMOTO CO., INC. (JP) 2013-08-01 US disclosed
US-20120136176-A1 CATALYST FOR ASYMMETRIC HYDROGENATION AND METHOD FOR MANUFACTURING OPTICALLY ACTIVE CARBONYL COMPOUND USING THE SAME TAKASAGO INTERNATIONAL CORPORATION (JP) 2012-05-31 US disclosed
US-7919468-B2 Compounds useful as modulators of the proteasome activity CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (C.N.R.S.) (FR) 2011-04-05 US disclosed
CN-101932560-A Matrix metalloproteinase inhibitors, pharmaceutical compositions containing them and their use POISON MED INST PLA MED ACAD 2010-12-29 CN disclosed
US-20090069222-A1 Compounds Useful as Modulators of the Proteasome Activity CENTRE NATIONAL DE AL RECHERCHE SCIENTIFIQUE (FR) 2009-03-12 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20130196050-A1 SALTY TASTE ENHANCER TAS2R10, TAS2R5, TAS1R1 MEN1 2795/4885KMT2A 1560/4885MAPT 4279/4885
US-20120136176-A1 CATALYST FOR ASYMMETRIC HYDROGENATION AND METHOD FOR MANUFACTURING OPTICALLY ACTIVE CARBONYL COMPOUND USING THE SAME HMOX1, HIRA, HRH1 MEN1 660/4885KMT2A 3823/4885MAPT 1810/4885
US-20090069222-A1 Compounds Useful as Modulators of the Proteasome Activity PSMB10, PSMB11, PSMB6 MEN1 2013/4885KMT2A 2725/4885MAPT 3169/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.