SCHEMBL9630702

SCHEMBL9630702

O=COC(=O)c1ccc(F)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
CA1 P00915 2/20 0.46
CA2 P00918 2/20 0.46
NPC1 O15118 5/20 0.46
RAB9A P51151 5/20 0.46
MAPT P10636 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
ATM Q13315 1/20 0.44
BCL2L1 Q07817 1/20 0.43
BAD Q92934 1/20 0.43
PKM P14618 1/20 0.43
TNFRSF1A P19438 1/20 0.42
CYP1A2 P05177 1/20 0.42
KDM4E B2RXH2 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
PLA2G7 Q13093 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2402587 0.89 ALDH1A1 (0.46) CA1CA2MAPTMEN1KMT2A
Fluorobenzene SCHEMBL28196684 0.86 PLA2G7 (0.50) CES2CES1NPC1RAB9AMAPT
SCHEMBL7868516 0.81 RAB9A (0.49) CES2CES1CA1CA2NPC1
SCHEMBL2835113 0.81 CES2 (0.48) CES2CES1CA1CA2NPC1
SCHEMBL593134 0.80 CA1 (0.56) CA1CA2MAPTMEN1KMT2A
SCHEMBL22191623 0.80 TSHR (0.55) CES2CES1CA1CA2MAPT
SCHEMBL248548 0.79 CES2 (0.62) CES2CES1CA1CA2NPC1
SCHEMBL15846817 0.78 LMNA (0.52) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL9364286 0.78 CES2 (0.50) CES2CES1CA1CA2NPC1
SCHEMBL10050028 0.78 TDP1 (0.59) CES2CES1NPC1RAB9AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-111333560-B Method for preparing spiro beta-lactam 合肥工业大学 2024-01-23 CN disclosed
CN-114409602-A Method for synthesizing alpha-keto acid by using oxalyl chloride and Grignard reagent as raw materials 武汉大学 2022-04-29 CN disclosed
CN-105330628-B Method for preparing 4-hydroxy butenolide from keto acid and alkyne 苏州大学 2021-10-26 CN disclosed
CN-106279023-B 3,4, 5-trisubstituted pyrazole compound, preparation method, pharmaceutical composition and application 中国科学院上海药物研究所 2021-06-22 CN disclosed
CN-107337581-B Process for preparing difluoroalcohol compounds 三和涂料工业有限公司 2020-12-29 CN disclosed
CN-111978201-A Synthesis method of N, N' -diaryl benzoyl hydrazine compound 甘肃农业大学 2020-11-24 CN disclosed
CN-108017635-A A kind of method of successive reaction synthesizing aryl benzoquinolizine ketone compounds 黑龙江大学 2018-05-11 CN disclosed
CN-107337581-A The method for preparing two fluoro alcoholic compounds 三和涂料工业有限公司 2017-11-10 CN disclosed
US-5140009-A Stable against proteolytic enzymes; anticarcinogenic agents; urogenital disorders TAP PHARMACEUTICALS, INC. (US) 1992-08-18 US disclosed
EP-0480918-A1 REDUCED SIZE LHRH ANALOGS ABBOTT LABORATORIES (US) 1992-04-22 EP disclosed
EP-0480918-A4 REDUCED SIZE LHRH ANALOGS. ABBOTT LAB (US) 1991-06-04 EP disclosed
EP-0417454-A2 Reduced size LHRH analogs ABBOTT LABORATORIES (US) 1991-03-20 EP disclosed
WO-1989007451-A1 REDUCED SIZE LHRH ANALOGS ABBOTT LABORATORIES (US) 1989-08-24 WO disclosed
EP-0328089-A2 Reduced size LHRH analogs ABBOTT LABORATORIES (US) 1989-08-16 EP disclosed
US-4255594-A Hydrogenation of halogen-containing carboxylic anhydrides ALLIED CHEMICAL CORPORATION (US) 1981-03-10 US disclosed