SCHEMBL9682042

SCHEMBL9682042

CCOC(=O)CCCSc1nc2ncccc2n1Cc1ccc(Cl)cc1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 4/20 0.53
DRD2 P14416 6/20 0.45
TBXA2R P21731 6/20 0.45
ALDH1A1 P00352 1/20 0.43
ATM Q13315 1/20 0.43
P2RX3 P56373 3/20 0.43
SLC22A12 Q96S37 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9681428 0.86 PTGDR2 (0.71) PTGDR2DRD2TBXA2RL3MBTL1
SCHEMBL9681251 0.86 L3MBTL1 (0.53) PTGDR2DRD2TBXA2RSLC22A12L3MBTL1
SCHEMBL9700228 0.86 ALDH1A1 (0.60) PTGDR2TBXA2RALDH1A1ATM
SCHEMBL9581575 0.79 TBXA2R (0.58) PTGDR2DRD2TBXA2RNPSR1
SCHEMBL9771980 0.77 P2RX3 (0.43) PTGDR2ALDH1A1P2RX3L3MBTL1NPSR1
SCHEMBL9699174 0.77 PTGDR2 (0.55) PTGDR2DRD2TBXA2RALDH1A1P2RX3
SCHEMBL9682472 0.77 TBXA2R (0.57) PTGDR2DRD2TBXA2R
SCHEMBL9699191 0.75 PTGDR2 (0.66) PTGDR2DRD2TBXA2RL3MBTL1NPSR1
SCHEMBL9683101 0.74 TBXA2R (0.56) TBXA2RP2RX3
SCHEMBL10386971 0.72 ALDH1A1 (0.57) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5128359-A Benzimidazole and azabenzimidazole derivatives which are thromboxane receptor antagonists, their methods of preparation LABORATOIRES UPSA (FR) 1992-07-07 US disclosed
US-5021443-A Noval benzimidazole and azabenzimiazole derivatives which are thromboxane receptor antagonists, their methods of preparation and pharmaceutical compositions in which they are present LABORATOIRES UPSA (FR) 1991-06-04 US disclosed