SCHEMBL9683479

SCHEMBL9683479

Nc1cc(Cl)ccc1NCc1ccc(Br)cc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1B1 P15121 2/20 0.43
TRAP1 Q12931 5/20 0.41
HSP90AA1 P07900 2/20 0.41
HSP90AB1 P08238 1/20 0.41
HSP90B1 P14625 3/20 0.39
BACE1 P56817 1/20 0.39
BACE2 Q9Y5Z0 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
LMNA P02545 1/20 0.38
MAPT P10636 1/20 0.38
HTT P42858 1/20 0.38
KDM1A O60341 1/20 0.38
AKR1A1 P14550 1/20 0.38
ADRA2B P18089 1/20 0.37
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
HPGD P15428 1/20 0.36
CYP2C19 P33261 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9683520 0.90 TRPM5 (0.43) AKR1B1MEN1KMT2AADRA2BALDH1A1
SCHEMBL9681422 0.86 HDAC1 (0.40) AKR1B1TRAP1HSP90B1MAPTKDM1A
SCHEMBL9682901 0.78 MAPT (0.43) AKR1B1MEN1KMT2AMAPTALDH1A1
SCHEMBL9682449 0.77 TRAP1 (0.44) AKR1B1TRAP1HSP90AA1HSP90AB1HSP90B1
SCHEMBL7746178 0.76 AKR1B1 (0.66) AKR1B1KMT2ALMNAMAPTAKR1A1
SCHEMBL9681992 0.75 HDAC8 (0.42) MEN1KMT2AMAPTL3MBTL1
SCHEMBL25828139 0.74 PTGER4 (0.56) LMNAMAPTHTTALDH1A1CYP1A2
SCHEMBL23630649 0.72 MAPT (0.44) MEN1KMT2ALMNAMAPTL3MBTL1
SCHEMBL11569274 0.72 ALDH1A1 (0.49) MEN1KMT2AMAPTALDH1A1HPGD
SCHEMBL6744214 0.72 ALDH1A1 (0.42) ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5128359-A Benzimidazole and azabenzimidazole derivatives which are thromboxane receptor antagonists, their methods of preparation LABORATOIRES UPSA (FR) 1992-07-07 US disclosed
US-5124336-A Cardiovascular disorders LABORATOIRES UPSA (FR) 1992-06-23 US disclosed