SCHEMBL9687928

SCHEMBL9687928

CCn1c(C(=O)OC(=O)c2cc3cc(NC(=O)OCc4ccccc4)ccc3[nH]2)cc2cc(NC(=O)OCc3ccccc3)ccc21

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MMP13 P45452 2/20 0.46
ROCK2 O75116 2/20 0.43
MGLL Q99685 2/20 0.41
MMP2 P08253 1/20 0.41
ALDH1A1 P00352 2/20 0.40
RAB9A P51151 2/20 0.40
NPC1 O15118 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
TSHR P16473 1/20 0.40
ATM Q13315 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
KDM4E B2RXH2 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C9 P11712 1/20 0.39
HPGD P15428 1/20 0.39
SRD5A2 P31213 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ADORA2B P29275 2/20 0.39
ADORA3 P0DMS8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9687922 0.90 SRD5A2 (0.46) MMP13ROCK2MGLLALDH1A1RAB9A
SCHEMBL8985820 0.82 MMP13 (0.68) MMP13ROCK2MGLLMMP2ALDH1A1
SCHEMBL8985906 0.79 SRD5A2 (0.60) MMP13ROCK2MGLLALDH1A1RAB9A
SCHEMBL9688119 0.77 MMP13 (0.61) MMP13ROCK2MGLLMMP2ALDH1A1
SCHEMBL7833243 0.75 LEF1 (0.55) MMP13ROCK2MGLLMMP2ALDH1A1
SCHEMBL5200855 0.71 MGLL (0.60) ROCK2MGLLALDH1A1RAB9ANPC1
SCHEMBL7908588 0.70 KCNQ2 (0.57) ROCK2MGLLALDH1A1RAB9ANPC1
SCHEMBL9127299 0.69 NPC1 (0.67) ALDH1A1RAB9ANPC1SMN1; SMN2KDM4E
SCHEMBL6741064 0.69 KDM4E (0.56) MMP13MMP2ALDH1A1RAB9ANPC1
SCHEMBL4432278 0.67 MGLL (0.65) ROCK2MGLLALDH1A1RAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0507861-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS. UPJOHN CO (US) 1992-10-14 EP disclosed
WO-1991009849-A1 DIAROMATIC SUBSTITUTED ANTI-AIDS COMPOUNDS THE UPJOHN COMPANY (US) 1991-07-11 WO disclosed