SCHEMBL9697283

SCHEMBL9697283

CC1(N2CCN(c3ccccn3)CC2)CN(c2ccccc2)c2ccccc2O1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 1/20 0.41
MEN1 O00255 3/20 0.40
KMT2A Q03164 3/20 0.40
NPSR1 Q6W5P4 1/20 0.40
MAPT P10636 3/20 0.38
ALDH1A1 P00352 2/20 0.38
KDM4E B2RXH2 2/20 0.38
OGA O60502 1/20 0.38
BCHE P06276 1/20 0.38
ACHE P22303 1/20 0.38
BACE1 P56817 1/20 0.38
DRD4 P21917 1/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
MAPK1 P28482 1/20 0.37
HTT P42858 1/20 0.37
PLD1 Q13393 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9530838 0.88 L3MBTL1 (0.46) KCNH2MAPTALDH1A1KDM4EACHE
SCHEMBL9530054 0.86 SIGMAR1 (0.39) MEN1KMT2AMAPTALDH1A1DRD4
SCHEMBL9455127 0.79 DRD2 (0.46) MEN1KMT2AMAPTALDH1A1KDM4E
SCHEMBL9529274 0.78 ALDH1A1 (0.43) MEN1KMT2AMAPTALDH1A1LMNA
SCHEMBL9530276 0.78 MAPT (0.45) KMT2ANPSR1MAPTALDH1A1DRD4
SCHEMBL9455326 0.72 L3MBTL1 (0.47) MEN1KMT2ANPSR1MAPTALDH1A1
SCHEMBL2627031 0.72 GRM5 (0.40) MEN1KMT2AALDH1A1POLB
SCHEMBL9529716 0.70 KCNH2 (0.50) KCNH2DRD4POLB
SCHEMBL9455304 0.70 OPRM1 (0.43) MAPTKDM4EDRD4LMNATP53
Hydrochloric Acid SCHEMBL9455139 0.69 CCR3 (0.43) MEN1KMT2ANPSR1KDM4EDRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5084454-A Tranquilizers and antinausea drugs FARMITALIA CARLO ERBA S.R.L. (IT) 1992-01-28 US disclosed
EP-0359790-A1 1,4-BENZOXAZINE AND 1,4-BENZOTHIAZINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION. ERBA CARLO SPA (IT) 1990-03-28 EP disclosed
WO-1989007596-A1 NEW 1,4-BENZOXAZINE AND 1,4-BENZOTHIAZINE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.R.L. (IT) 1989-08-24 WO disclosed