SCHEMBL9707504

SCHEMBL9707504

Cc1nc2c(c(=O)n(-c3ccccc3)c(=O)n2C)n1Cc1ccc(-c2ccccc2-c2nnn[nH]2)cc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
ALOX15 P16050 1/20 0.39
HSD17B10 Q99714 1/20 0.39
LMNA P02545 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HTT P42858 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
AGTR1 P30556 2/20 0.38
AGTR2 P50052 2/20 0.38
MAPT P10636 1/20 0.38
BRAF P15056 1/20 0.38
PIK3CG P48736 1/20 0.38
POLB P06746 1/20 0.38
PCSK9 Q8NBP7 1/20 0.38
DPP4 P27487 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9707766 0.93 ALDH1A1 (0.42) ALDH1A1ALOX15HSD17B10LMNASMN1; SMN2
SCHEMBL9707935 0.93 AGTR1 (0.39) ALDH1A1AGTR1AGTR2
SCHEMBL9708509 0.91 ADORA3 (0.40) AGTR1AGTR2
SCHEMBL9707722 0.91 AGTR1 (0.39) ALDH1A1AGTR1AGTR2
SCHEMBL9708711 0.90 ALOX15 (0.46) ALDH1A1ALOX15HSD17B10LMNASMN1; SMN2
SCHEMBL9708369 0.90 AGTR1 (0.39) AGTR1AGTR2
SCHEMBL9707431 0.90 ALDH1A1 (0.44) ALDH1A1ALOX15HSD17B10SMN1; SMN2HTT
SCHEMBL9708188 0.89 USP1 (0.39) ALDH1A1ALOX15HSD17B10LMNASMN1; SMN2
SCHEMBL9707609 0.89 DCTPP1 (0.40) ALDH1A1SMN1; SMN2AGTR1AGTR2
SCHEMBL9708087 0.88 ADORA1 (0.38) AGTR1AGTR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992007852-A1 BIPHENYLALKYL XANTHINE COMPOUNDS FOR TREATMENT OF CARDIOVASCULAR DISORDERS G.D. SEARLE & CO. (US) 1992-05-14 WO disclosed