SCHEMBL9714916

SCHEMBL9714916

Cc1ccc(-c2[nH]nc(N(C)C)c2CC(=O)N(C)C)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.41
GABRA1 P14867 3/20 0.41
GABRB2 P47870 3/20 0.41
KDM4E B2RXH2 1/20 0.41
ALB P02768 1/20 0.41
CYP3A4 P08684 1/20 0.41
CHRM1 P11229 1/20 0.41
HPGD P15428 1/20 0.41
GABRB1 P18505 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA3 P34903 1/20 0.41
ADRA1A P35348 1/20 0.41
OPRK1 P41145 1/20 0.41
HTR2B P41595 1/20 0.41
GABRA2 P47869 1/20 0.41
KCNH2 Q12809 1/20 0.41
HSD17B10 Q99714 1/20 0.41
ALPL P05186 1/20 0.35
TSPO P30536 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9714971 0.87 TSPO (0.46) TSPO
Hydrochloric Acid SCHEMBL9714930 0.86 LMNA (0.41) LMNAKDM4EALPLTYMP
SCHEMBL9715039 0.84 LMNA (0.42) LMNAKDM4EHPGDHSD17B10ALPL
SCHEMBL9714924 0.78 HSD17B10 (0.41) LMNAKDM4ECYP3A4HPGDHSD17B10
SCHEMBL9715021 0.78 PTGDR2 (0.39) KDM4EHPGDALPLTSPOSMN1; SMN2
Hydrochloric Acid SCHEMBL9714965 0.78 RAB9A (0.53) LMNAKDM4EHPGDHSD17B10ALPL
Hydrochloric Acid SCHEMBL9714991 0.78 HSD17B10 (0.40) LMNAKDM4ECYP3A4HPGDHSD17B10
Hydrochloric Acid SCHEMBL9715064 0.77 PTGDR2 (0.39) KDM4EHPGDALPLTSPOSMN1; SMN2
SCHEMBL9714951 0.75 P2RX7 (0.39) KDM4ETSPOSMN1; SMN2
Hydrochloric Acid SCHEMBL9714943 0.69 L3MBTL1 (0.45) KDM4ECYP3A4HPGDHSD17B10SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992018484-A1 3-AMINO-5-ARYLPYRAZOLE-4-ACETIC ACID DERIVATIVES EXHIBITING THERAPEUTIC EFFECTS A.H. ROBINS COMPANY, INCORPORATED (US) 1992-10-29 WO claimed
US-5057534-A Anxiolytic, anticonfulsant and muscle relaxants A. H. ROBINS COMPANY INCORPORATED (US) 1991-10-15 US claimed
WO-1992018484-A1 3-AMINO-5-ARYLPYRAZOLE-4-ACETIC ACID DERIVATIVES EXHIBITING THERAPEUTIC EFFECTS A.H. ROBINS COMPANY, INCORPORATED (US) 1992-10-29 WO disclosed