SCHEMBL9728783

SCHEMBL9728783

N#Cc1sc(N)nc1C1=CCCN(CCc2ccccc2)C1

nearest known ligand 0.60

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
MEN1 O00255 1/20 0.46
ALDH1A1 P00352 1/20 0.46
GLA P06280 1/20 0.46
GAA P10253 1/20 0.46
MAPT P10636 1/20 0.46
KMT2A Q03164 1/20 0.46
TAAR1 Q96RJ0 1/20 0.46
MAOA P21397 1/20 0.37
CHRM1 P11229 1/20 0.37
NOS3 P29474 1/20 0.36
NOS1 P29475 1/20 0.36
GRM2 Q14416 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9728276 0.90 MAOA (0.39) KDM4EMEN1ALDH1A1GLAGAA
Hydrochloric Acid SCHEMBL9728481 0.85 SIGMAR1 (0.46)
SCHEMBL9729439 0.84 MAOA (0.39) KDM4EMEN1ALDH1A1GLAGAA
SCHEMBL9728560 0.81
SCHEMBL9729054 0.81 RAD52 (0.40) KDM4EMEN1ALDH1A1GAAMAPT
Hydrochloric Acid SCHEMBL9729647 0.76 CHRM1 (0.44) CHRM1
SCHEMBL9451990 0.75 ALDH1A1 (0.46) ALDH1A1MAPTKMT2ATAAR1
SCHEMBL9728485 0.73 DRD2 (0.43) MEN1ALDH1A1GAAKMT2A
SCHEMBL9728509 0.69 THRB (0.39)
SCHEMBL1449744 0.66 CDC7 (0.58) KDM4EALDH1A1GLAGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5128340-A Thiazole derivatives AKZO N.V. (NL) 1992-07-07 US disclosed
EP-0368384-A1 Thiazole derivatives AKZO N.V. (NL) 1990-05-16 EP disclosed