SCHEMBL9732964

SCHEMBL9732964

COc1cccn(C2=CC(C)(C)Cc3ccc(C#N)cc32)c1=O

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.35
DRD4 P21917 1/20 0.35
DRD3 P35462 1/20 0.35
GSK3B P49841 2/20 0.33
ALK Q9UM73 2/20 0.33
STK10 O94804 1/20 0.33
CLK2 P49760 1/20 0.33
GSK3A P49840 1/20 0.33
SLK Q9H2G2 1/20 0.33
CLK4 Q9HAZ1 1/20 0.33
ICMT O60725 1/20 0.33
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
AR P10275 1/20 0.33
PGR P06401 1/20 0.33
CECR2 Q9BXF3 1/20 0.33
BACE1 P56817 1/20 0.33
KDM1A O60341 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733300 0.88 MAOB (0.32) ALKPGR
SCHEMBL9733746 0.85 PGR (0.34) ICMTPGRBACE1
SCHEMBL9733259 0.85 PGR (0.34) PGRBACE1
SCHEMBL9734356 0.85 POLB (0.34) ALKPGRBACE1
SCHEMBL9733975 0.82 KCNH2 (0.37) ALKPGRMAPT
SCHEMBL9733088 0.82 MAPT (0.36) ALKARPGRMAPT
SCHEMBL9733284 0.81 HTR1A (0.37) GSK3BPGRBACE1CCNB2CDK1
SCHEMBL9733001 0.80 OTUD7B (0.35) DRD2DRD3ALKPGRBACE1
SCHEMBL7267589 0.79 PDE4A (0.49) GSK3BALKSTK10CLK2GSK3A
SCHEMBL9733106 0.79 PGR (0.34) ALKPDE4APGRBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US disclosed
EP-0368160-A1 Tetralin derivatives MERCK PATENT GmbH (DE) 1990-05-16 EP disclosed