SCHEMBL9733106

SCHEMBL9733106

CC1(C)C=C(n2cccnc2=O)c2cc(C#N)ccc2C1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PGR P06401 1/20 0.34
PDE4A P27815 2/20 0.33
CYP11B2 P19099 3/20 0.33
SLC11A2 P49281 1/20 0.33
CYP11B1 P15538 1/20 0.32
ALK Q9UM73 1/20 0.32
BACE1 P56817 3/20 0.32
DDB1 Q16531 1/20 0.32
CRBN Q96SW2 1/20 0.32
GABRA1 P14867 1/20 0.32
GABRG2 P18507 1/20 0.32
GABRB3 P28472 1/20 0.32
GABRA5 P31644 1/20 0.32
GABRA3 P34903 1/20 0.32
GABRA2 P47869 1/20 0.32
NSD2 O96028 1/20 0.32
POLB P06746 1/20 0.32
CASP3 P42574 1/20 0.32
HTR2C P28335 1/20 0.32
GRM5 P41594 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733284 0.83 HTR1A (0.37) PGRBACE1GABRA1GABRG2GABRB3
SCHEMBL9733759 0.82 TDP2 (0.35) PGRCYP11B2BACE1POLBCASP3
SCHEMBL9734356 0.80 POLB (0.34) PGRALKBACE1NSD2POLB
SCHEMBL9733774 0.80 HTR1A (0.38) PGRCYP11B2CYP11B1BACE1POLB
SCHEMBL9733746 0.80 PGR (0.34) PGRBACE1NSD2POLBCASP3
SCHEMBL9733259 0.80 PGR (0.34) PGRCYP11B2BACE1NSD2POLB
SCHEMBL9733957 0.79 CYP19A1 (0.35) PGRCYP11B2CYP11B1BACE1POLB
SCHEMBL9732964 0.79 DRD2 (0.35) PGRPDE4AALKBACE1
SCHEMBL9733966 0.79 ALDH1A1 (0.33) PGR
SCHEMBL8085075 0.78 PDE4A (0.41) PDE4ADDB1CRBNCASP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US disclosed
EP-0368160-A1 Tetralin derivatives MERCK PATENT GmbH (DE) 1990-05-16 EP disclosed