SCHEMBL9733488

SCHEMBL9733488

CC(c1c(F)cccc1F)c1nnc(C(N)=O)n1C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 3/20 0.37
CA5A P35218 1/20 0.35
CES2 O00748 1/20 0.33
CES1 P23141 1/20 0.33
RIPK1 Q13546 1/20 0.33
MAPT P10636 3/20 0.32
ALDH1A1 P00352 2/20 0.32
NR1I2 O75469 1/20 0.32
AHR P35869 1/20 0.32
MC4R P32245 1/20 0.32
MET P08581 3/20 0.31
TP53 P04637 1/20 0.31
PARP1 P09874 1/20 0.30
MEN1 O00255 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP3A4 P08684 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30
CYP2C19 P33261 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9735004 0.70 CA5A (0.44) CA5AALDH1A1TP53
SCHEMBL9733462 0.68 GAA (0.48) ALDH1A1MEN1KMT2ANPSR1
SCHEMBL29718627 0.65 CES2 (0.46) CES2CES1ALDH1A1MEN1KMT2A
SCHEMBL20970373 0.64 IRAK4 (0.43) CES2CES1MAPTALDH1A1PARP1
SCHEMBL13572952 0.64 KDM4E (0.45) MAPTALDH1A1MEN1CYP2D6KMT2A
SCHEMBL10959131 0.64 CA5A (0.52) CA5ACES2CES1ALDH1A1NPSR1
SCHEMBL9714322 0.61 ADA (0.48) CA5ACES2CES1
SCHEMBL9714477 0.61 ALDH1A1 (0.49) CES2CES1ALDH1A1CYP1A2CYP3A4
SCHEMBL21066343 0.60 GAA (0.35) ALDH1A1TP53
SCHEMBL10403668 0.60 DAPK3 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5098922-A Anticonvulsants CIBA-GEIGY CORPORATION (US) 1992-03-24 US claimed
US-5045556-A Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY CORPORATION (US) 1991-09-03 US claimed
EP-0267147-B1 ARALKYL-4H-1,2,4-TRIAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-07 EP claimed
EP-0267147-A1 Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY AG (CH) 1988-05-11 EP claimed
US-5098922-A Anticonvulsants CIBA-GEIGY CORPORATION (US) 1992-03-24 US disclosed
US-5045556-A Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY CORPORATION (US) 1991-09-03 US disclosed
EP-0267147-B1 ARALKYL-4H-1,2,4-TRIAZOLE DERIVATIVES CIBA-GEIGY AG (CH) 1991-08-07 EP disclosed
EP-0267147-A1 Aralkyl-4H-1,2,4-triazole derivatives CIBA-GEIGY AG (CH) 1988-05-11 EP disclosed