SCHEMBL9733759

SCHEMBL9733759

CC1(C)C=C(n2ccc(O)nc2=O)c2cc(C#N)ccc2C1

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
TDP2 O95551 1/20 0.35
BACE1 P56817 1/20 0.32
PGR P06401 1/20 0.31
POLB P06746 1/20 0.31
CASP3 P42574 1/20 0.31
CYP11B2 P19099 2/20 0.31
MALT1 Q9UDY8 1/20 0.30
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
KDM4C Q9H3R0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733622 0.84 POLB (0.35) TDP2BACE1PGRPOLBCASP3
SCHEMBL9734020 0.82 CYP11B2 (0.37) BACE1PGRPOLBCASP3CYP11B2
SCHEMBL9733106 0.82 PGR (0.34) BACE1PGRPOLBCASP3CYP11B2
SCHEMBL9733259 0.80 PGR (0.34) BACE1PGRPOLBCASP3CYP11B2
SCHEMBL7275951 0.79 PDE4A (0.41) TDP2CASP3MALT1
SCHEMBL9733851 0.78 MAOB (0.34) TDP2BACE1PGRPOLBCASP3
SCHEMBL9733284 0.78 HTR1A (0.37) BACE1PGRPOLBCASP3
SCHEMBL9733774 0.77 HTR1A (0.38) BACE1PGRPOLBCASP3CYP11B2
SCHEMBL9733886 0.77 PGR (0.34) BACE1PGRPOLBCASP3CYP11B2
SCHEMBL9733957 0.76 CYP19A1 (0.35) BACE1PGRPOLBCASP3CYP11B2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US disclosed
EP-0368160-A1 Tetralin derivatives MERCK PATENT GmbH (DE) 1990-05-16 EP disclosed