SCHEMBL9733622

SCHEMBL9733622

CC1(C)C=C(n2ccc(O)cc2=O)c2cc(C#N)ccc2C1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.35
MAOB P27338 3/20 0.34
MAOA P21397 2/20 0.34
PGR P06401 2/20 0.33
CASP3 P42574 1/20 0.33
MALT1 Q9UDY8 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
MIF P14174 1/20 0.32
BACE1 P56817 1/20 0.31
SIGMAR1 Q99720 1/20 0.31
NSD2 O96028 1/20 0.30
ABCC9 O60706 2/20 0.30
ABCC8 Q09428 2/20 0.30
KCNJ11 Q14654 2/20 0.30
KCNJ8 Q15842 2/20 0.30
TDP2 O95551 1/20 0.30
CYP1A2 P05177 1/20 0.30
CYP2D6 P10635 1/20 0.30
CYP2C9 P11712 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733851 0.85 MAOB (0.34) POLBMAOBMAOAPGRCASP3
SCHEMBL9733284 0.85 HTR1A (0.37) POLBPGRCASP3BACE1NSD2
SCHEMBL10433117 0.84 ESR1 (0.34) POLBMAOBMAOATDP2
SCHEMBL9733759 0.84 TDP2 (0.35) POLBPGRCASP3MALT1HTR2A
SCHEMBL9733774 0.82 HTR1A (0.38) POLBPGRCASP3BACE1ABCC9
SCHEMBL9734020 0.82 CYP11B2 (0.37) POLBMAOBMAOAPGRCASP3
SCHEMBL9733259 0.82 PGR (0.34) POLBPGRCASP3MALT1HTR2A
SCHEMBL9733645 0.81 GAA (0.37) PGRCASP3TDP2CYP2C9CYP2C19
SCHEMBL9733222 0.79 POLB (0.34) POLBPGRCASP3MALT1HTR2A
SCHEMBL9735211 0.79 ABCC9 (0.34) POLBPGRCASP3MALT1HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US claimed
EP-0368160-A1 Tetralin derivatives MERCK PATENT GmbH (DE) 1990-05-16 EP claimed
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US disclosed
EP-0368160-A1 Tetralin derivatives MERCK PATENT GmbH (DE) 1990-05-16 EP disclosed