SCHEMBL9733774

SCHEMBL9733774

CC1(C)C=C(n2ccncc2=O)c2cc(C#N)ccc2C1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.38
CYP11B2 P19099 10/20 0.36
CYP11B1 P15538 9/20 0.36
ABCC9 O60706 1/20 0.35
CYP19A1 P11511 1/20 0.35
PGR P06401 1/20 0.32
BACE1 P56817 1/20 0.32
POLB P06746 1/20 0.32
CASP3 P42574 1/20 0.32
GSK3A P49840 1/20 0.31
GSK3B P49841 1/20 0.31
CDK5 Q00535 1/20 0.31
CDK5R1 Q15078 1/20 0.31
GRM5 P41594 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9733957 0.83 CYP19A1 (0.35) CYP11B2CYP11B1ABCC9CYP19A1PGR
SCHEMBL9733284 0.83 HTR1A (0.37) HTR1AABCC9PGRBACE1POLB
SCHEMBL9733622 0.82 POLB (0.35) ABCC9PGRBACE1POLBCASP3
SCHEMBL9733106 0.80 PGR (0.34) CYP11B2CYP11B1PGRBACE1POLB
SCHEMBL8085306 0.78 ABCC9 (0.41) HTR1ACYP11B2CYP11B1ABCC9CASP3
SCHEMBL9734020 0.78 CYP11B2 (0.37) CYP11B2PGRBACE1POLBCASP3
SCHEMBL9733759 0.77 TDP2 (0.35) CYP11B2PGRBACE1POLBCASP3
SCHEMBL9733851 0.77 MAOB (0.34) ABCC9PGRBACE1POLBCASP3
SCHEMBL9735211 0.77 ABCC9 (0.34) ABCC9PGRPOLBCASP3
SCHEMBL9733784 0.77 CYP11B2 (0.35) CYP11B2CYP11B1ABCC9PGRBACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5132307-A TETRALIN COMPOUNDS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1992-07-21 US disclosed