SCHEMBL9737185

SCHEMBL9737185

CNC(=O)Cc1c(-c2ccc(C)cc2)nn2cccnc12

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
KCNQ3 O43525 10/20 0.41
KCNQ2 O43526 10/20 0.41
MYC P01106 1/20 0.41
PTGS2 P35354 1/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
HPGD P15428 1/20 0.38
HSD17B10 Q99714 1/20 0.38
PLK1 P53350 1/20 0.37
DPP4 P27487 1/20 0.37
IRAK4 Q9NWZ3 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9737626 0.91 KCNQ3 (0.45) KCNQ3KCNQ2MYCPTGS2KDM4E
SCHEMBL9738434 0.90 KCNQ3 (0.41) KCNQ3KCNQ2MYCPTGS2ALDH1A1
SCHEMBL9737283 0.87 PTGDR2 (0.47) MYCPTGS2KDM4EALDH1A1
SCHEMBL9737491 0.86 PTGS2 (0.41) KCNQ3KCNQ2MYCPTGS2KDM4E
SCHEMBL9737572 0.84 TSPO (0.45) KCNQ3KCNQ2MYCPTGS2KDM4E
SCHEMBL9737163 0.83 ALDH1A1 (0.43) MYCPTGS2KDM4EALDH1A1HPGD
SCHEMBL9738542 0.81 TSPO (0.44)
SCHEMBL9737222 0.80 MYC (0.39) KCNQ3KCNQ2MYCPTGS2ALDH1A1
SCHEMBL9737699 0.76 PTGDR2 (0.46) KCNQ3KCNQ2PTGS2KDM4EALDH1A1
SCHEMBL9737634 0.75 KDM4E (0.48) KDM4EALDH1A1CYP1A2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5114944-A Anxiolytic and anticonvulsant agents; muscle relaxants A. H. ROBINS COMPANY INCORPORATED (US) 1992-05-19 US claimed
US-5114944-A Anxiolytic and anticonvulsant agents; muscle relaxants A. H. ROBINS COMPANY INCORPORATED (US) 1992-05-19 US disclosed