SCHEMBL9211609

SCHEMBL9211609

Cc1cccc(OCCCN2CCCC(COS(=O)(=O)c3ccccc3)C2)c1

nearest known ligand 0.55

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.55
L3MBTL1 Q9Y468 1/20 0.55
HTR1A P08908 1/20 0.52
HTR7 P34969 1/20 0.52
HRH3 Q9Y5N1 8/20 0.49
ALDH1A1 P00352 2/20 0.47
KMT2A Q03164 1/20 0.47
HRH2 P25021 1/20 0.45
HRH1 P35367 1/20 0.45
DRD2 P14416 1/20 0.44
DRD1 P21728 1/20 0.44
DRD4 P21917 1/20 0.44
DRD5 P21918 1/20 0.44
DRD3 P35462 1/20 0.44
CHRNB2 P17787 1/20 0.43
CHRNB4 P30926 1/20 0.43
CHRNA3 P32297 1/20 0.43
CHRNA4 P43681 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9740303 0.91 HRH3 (0.60) KDM4EHRH3ALDH1A1KMT2ACHRNB2
SCHEMBL9739220 0.86 HRH3 (0.52) KDM4EHRH3ALDH1A1KMT2ADRD3
SCHEMBL9739552 0.86 CHRNB2 (0.57) KDM4EHRH3ALDH1A1KMT2AHRH2
SCHEMBL9740276 0.80 HTR1A (0.52) KDM4EL3MBTL1HTR1AHTR7HRH3
SCHEMBL9208504 0.80 HRH2 (0.49) KDM4EHRH3ALDH1A1KMT2AHRH2
SCHEMBL9205099 0.79 HRH3 (0.48) KDM4EHRH3ALDH1A1KMT2ADRD4
SCHEMBL9210505 0.79 HRH3 (0.57) KDM4EHRH3ALDH1A1KMT2ACHRNB2
SCHEMBL9215679 0.77 KDM4E (0.67) KDM4EL3MBTL1HRH3ALDH1A1KMT2A
SCHEMBL9212384 0.74 ADRA1A (0.52) KDM4EHTR1AHTR7ALDH1A1KMT2A
SCHEMBL9205156 0.74 CHRNB2 (0.54) KDM4EHRH3ALDH1A1KMT2ACHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed