SCHEMBL9739485

SCHEMBL9739485

O=C1c2ccccc2C2(c3cccc4ncccc34)CCCN12

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.37
P2RX7 Q99572 2/20 0.37
TSHR P16473 2/20 0.37
CYP3A4 P08684 1/20 0.37
NFKB1 P19838 1/20 0.37
THPO P40225 1/20 0.37
HIF1A Q16665 1/20 0.37
MAPT P10636 3/20 0.37
SMN1; SMN2 Q16637 2/20 0.37
KDM4E B2RXH2 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
CASP1 P29466 1/20 0.37
HTT P42858 1/20 0.37
HBB P68871 1/20 0.37
KMT2A Q03164 1/20 0.37
CCNC P24863 1/20 0.36
CDK8 P49336 1/20 0.36
LMNA P02545 1/20 0.36
BLM P54132 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9740266 0.94 SLC22A12 (0.38) MAPTSMN1; SMN2MEN1ALDH1A1KMT2A
SCHEMBL9739249 0.82 SLC6A3 (0.40) MAPTSMN1; SMN2MEN1HTTKMT2A
SCHEMBL9738592 0.79 HSD11B1 (0.41) SMN1; SMN2MEN1HTTKMT2ANPC1
SCHEMBL9701851 0.78 TSHR (0.37) CYP1A2P2RX7TSHRCYP3A4NFKB1
SCHEMBL9739775 0.76 NPC1 (0.38) SMN1; SMN2HTTCCNCCDK8NPC1
SCHEMBL9740491 0.75 MEN1 (0.40) CYP1A2CYP3A4MAPTSMN1; SMN2MEN1
SCHEMBL9739705 0.75 MEN1 (0.37) CYP1A2MAPTSMN1; SMN2MEN1HTT
SCHEMBL9739157 0.75 PARP1 (0.39) MAPTSMN1; SMN2KDM4EMEN1ALDH1A1
SCHEMBL9738986 0.75 RXFP1 (0.42) CYP1A2TSHRCYP3A4SMN1; SMN2MEN1
SCHEMBL9740469 0.74 GAA (0.43) MAPTSMN1; SMN2KDM4EMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992016529-A1 NOVEL ISOINDOLE DERIVATIVES AND MEDICAMENTS CONTAINING THEM BOEHRINGER MANNHEIM GMBH (DE) 1992-10-01 WO disclosed