SCHEMBL9752900

SCHEMBL9752900

CC(C)(C)OC(=O)N[C@H](CCCC(N)=O)Sc1ccc2ccccc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX1 P07099 1/20 0.45
CTSK P43235 8/20 0.44
CTSB P07858 1/20 0.44
CTSS P25774 1/20 0.44
GABRB1 P18505 1/20 0.43
GABRB2 P47870 1/20 0.43
SIRT5 Q9NXA8 1/20 0.40
ACE P12821 1/20 0.38
HDAC4 P56524 2/20 0.38
HDAC1 Q13547 2/20 0.38
ACACB O00763 1/20 0.37
MMP13 P45452 1/20 0.37
KDM4A O75164 1/20 0.37
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC11 Q96DB2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9752897 0.76 CTSK (0.47) EPHX1CTSKCTSBCTSSGABRB1
SCHEMBL9753260 0.72 EPHX1 (0.41) EPHX1CTSKCTSBCTSSGABRB1
SCHEMBL16317891 0.72 PLA2G2A (0.45) CTSKCTSBCTSSGABRB1GABRB2
SCHEMBL24415818 0.72 GABRB1 (0.48) EPHX1CTSKCTSBCTSSGABRB1
SCHEMBL7289392 0.71 PPARA (0.57) CTSKCTSBCTSSGABRB1GABRB2
SCHEMBL5228193 0.71 PPARA (0.57) CTSKCTSBCTSSGABRB1GABRB2
SCHEMBL7250898 0.71 PPARA (0.57) CTSKCTSBCTSSGABRB1GABRB2
SCHEMBL7655882 0.70 CTSS (0.69) CTSKCTSBCTSSACEHDAC8
SCHEMBL9331930 0.70 CTSS (0.69) CTSKCTSBCTSSACEHDAC8
SCHEMBL8362256 0.70 GABRB1 (0.52) CTSKCTSBCTSSGABRB1GABRB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991008737-A2 PHARMACOLOGICALLY ACTIVE AMIDE CARBOXYLATE DERIVATIVES FISONS PLC (GB) 1991-06-27 WO disclosed