SCHEMBL9754633

SCHEMBL9754633

COC(=O)N(C(=O)[C@H](C)N)[C@@H](C)C(=O)NCC(C(=O)O)C(NCCCCCCc1ccccc1)C(=O)NC(C(=O)OCc1ccccc1)C(C)C

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
LNPEP Q9UIQ6 5/20 0.39
ERAP2 Q6P179 4/20 0.38
ERAP1 Q9NZ08 2/20 0.38
CA2 P00918 1/20 0.37
CA5A P35218 1/20 0.37
CTSB P07858 1/20 0.36
CTSK P43235 1/20 0.36
CA1 P00915 1/20 0.34
REN P00797 1/20 0.34
CTSD P07339 1/20 0.34
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.33
IL1RN P18510 1/20 0.33
CPB1 P15086 1/20 0.33
CPB2 Q96IY4 1/20 0.33
ITGB3 P05106 1/20 0.33
ITGAV P06756 1/20 0.33
ITGA2B P08514 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7332099 0.82 LNPEP (0.37) LNPEPERAP2ERAP1CA2CA5A
SCHEMBL7322813 0.76 CTSD (0.37) CA2CA5ACTSD
SCHEMBL7324031 0.75 CASP1 (0.38) CTSDALDH1A1CPB2
SCHEMBL9754438 0.73 ALOX5 (0.32) CA2CA5AALDH1A1MAPT
SCHEMBL9296616 0.72 CA2 (0.34) LNPEPERAP2ERAP1CA2CA5A
SCHEMBL7270142 0.70 CYP2D6 (0.51) ERAP2ERAP1CA2CA5AIL1RN
SCHEMBL7270146 0.70 CYP2D6 (0.51) ERAP2ERAP1CA2CA5AIL1RN
SCHEMBL7327734 0.68 ALOX5 (0.32) CA2CA5AALDH1A1MAPT
SCHEMBL10954138 0.68 ACE (0.45)
SCHEMBL10953109 0.68 LGMN (0.41) CTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1991015121-A1 METHOD FOR TREATING FUNGAL INFECTION SMITHKLINE BEECHAM CORPORATION (US) 1991-10-17 WO disclosed