SCHEMBL977421

SCHEMBL977421

CCCCCCCCC=CCCCCCCCC(=O)N(C(=O)CCCCCCCC=CCCCCCCCC)C(=O)OC(C)CN(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.47
FAAH O00519 4/20 0.45
TERT O14746 3/20 0.44
PTPN1 P18031 3/20 0.44
PPARG P37231 3/20 0.44
PPARD Q03181 3/20 0.44
PPARA Q07869 3/20 0.44
CYP1A2 P05177 2/20 0.44
MAPT P10636 2/20 0.44
CYP2C19 P33261 2/20 0.44
BLM P54132 2/20 0.44
HSD17B10 Q99714 2/20 0.44
FABP4 P15090 2/20 0.44
KMT2A Q03164 2/20 0.44
GMNN O75496 1/20 0.44
USP2 O75604 1/20 0.44
LMNA P02545 1/20 0.44
POLB P06746 1/20 0.44
CYP2C9 P11712 1/20 0.44
ALOX15 P16050 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19692318 1.00 EPHX2 (0.47) EPHX2FAAHTERTPTPN1PPARG
SCHEMBL465985 0.84 PRKCA (0.54) FAAHTERTCYP1A2MAPTCYP2C19
SCHEMBL992184 0.84 PRKCA (0.54) FAAHTERTCYP1A2MAPTCYP2C19
SCHEMBL31374704 0.81 ALDH1A1 (0.58) FAAHPPARGPPARDPPARAMAPT
SCHEMBL28450589 0.80 EPHX2 (0.50) EPHX2FAAHTERTPTPN1PPARG
SCHEMBL25140 0.79 ALDH1A1 (0.43) FAAHPPARGPPARDPPARAMAPT
SCHEMBL158797 0.77 ALDH1A1 (0.51) EPHX2PPARGPPARDPPARAHSD17B10
SCHEMBL10016290 0.77 TSHR (0.42) EPHX2PTPN1PPARGPPARACYP1A2
SCHEMBL15205542 0.77 TSHR (0.42) EPHX2PTPN1PPARGPPARACYP1A2
SCHEMBL6686505 0.77 TERT (0.66) EPHX2FAAHTERTPTPN1PPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 131 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12016929-B2 Lipid formulations for delivery of therapeutic agents ARBUTUS BIOPHARMA CORPORATION (CA) 2024-06-25 US disclosed
US-20240182895-A1 NON-LIPOSOMAL SYSTEMS FOR NUCLEIC ACID DELIVERY ARBUTUS BIOPHARMA CORPORATION (CA) 2024-06-06 US disclosed
US-20240148875-A1 NOVEL LIPID FORMULATIONS FOR DELIVERY OF THERAPEUTIC AGENTS ARBUTUS BIOPHARMA CORPORATION (CA) 2024-05-09 US disclosed
WO-2024073678-A2 PHOSPHOLIPIDS CONTAINING A HETEROCYCLE RING HAVING A TERTIARY AMINE OR AMIDE OMEGA THERAPEUTICS, INC. (US) 2024-04-04 WO disclosed
US-20240100166-A1 NOVEL LIPID FORMULATIONS FOR DELIVERY OF THERAPEUTIC AGENTS ARBUTUS BIOPHARMA CORPORATION (CA) 2024-03-28 US disclosed
EP-4328314-A2 LIPID NANOPARTICLE METHODS AND COMPOSITIONS FOR PRODUCING ENGINEERED ERYTHROID CELLS Tessera Therapeutics, Inc. (US) 2024-02-28 EP disclosed
US-11904052-B2 Methods for ameliorating infusion reactions ARBUTUS BIOPHARMA CORPORATION (CA) 2024-02-20 US disclosed
US-20240050463-A1 THERAPEUTIC COMPOSITIONS AND METHODS FOR TREATING HEPATITIS B ARBUTUS BIOPHARMA CORPORATION (US) 2024-02-15 US disclosed
US-20240035030-A1 NON-LIPOSOMAL SYSTEMS FOR NUCLEIC ACID DELIVERY ARBUTUS BIOPHARMA CORPORATION (CA) 2024-02-01 US disclosed
WO-2023225621-A2 LIPIDS FOR DELIVERY OF THERAPEUTIC AGENTS OMEGA THERAPEUTICS, INC. (US) 2023-11-23 WO disclosed
WO-2011141703-A1 COMPOSITIONS AND METHODS FOR SILENCING APOLIPOPROTEIN B PROTIVA BIOTHERAPEUTICS INC. (CA) 2011-11-17 WO disclosed
WO-2011141704-A1 NOVEL CYCLIC CATIONIC LIPIDS AND METHODS OF USE PROTIVA BIOTHERAPEUTICS, INC (CA) 2011-11-17 WO disclosed
WO-2011141705-A1 NOVEL CATIONIC LIPIDS AND METHODS OF USE THEREOF PROTIVA BIOTHERAPEUTICS, INC. (CA) 2011-11-17 WO disclosed
US-20110201667-A1 COMPOSITIONS AND METHODS FOR SILENCING EBOLA VIRUS GENE EXPRESSION PROTIVA BIOTHERAPEUTICS, INC. (CA) 2011-08-18 US disclosed
US-20110195127-A1 COMPOSITIONS AND METHODS FOR SILENCING APOLIPOPROTEIN B PROTIVA BIOTHERAPEUTICS, INC. (CA) 2011-08-11 US disclosed
US-20110117125-A1 COMPOSITIONS AND METHODS FOR THE DELIVERY OF NUCLEIC ACIDS TEKMIRA PHARMACEUTICALS CORPORATION (CA) 2011-05-19 US disclosed
US-20110076335-A1 NOVEL LIPID FORMULATIONS FOR DELIVERY OF THERAPEUTIC AGENTS TO SOLID TUMORS PROTIVA BIOTHERAPEUTICS, INC. (CA) 2011-03-31 US disclosed
WO-2011000106-A1 IMPROVED CATIONIC LIPIDS AND METHODS FOR THE DELIVERY OF THERAPEUTIC AGENTS PROTIVA BIOTHERAPEUTICS, INC. (CA) 2011-01-06 WO disclosed
WO-2011000107-A1 NOVEL LIPID FORMULATIONS FOR DELIVERY OF THERAPEUTIC AGENTS TO SOLID TUMORS PROTIVA BIOTHERAPEUTICS, INC. (CA) 2011-01-06 WO disclosed
WO-2011000108-A1 COMPOSITIONS AND METHODS FOR SILENCING APOLIPOPROTEIN B PROTIVA BIOTHERAPEUTICS, INC. (CA) 2011-01-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (11 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110076335-A1 NOVEL LIPID FORMULATIONS FOR DELIVERY OF THERAPEUTIC AGENTS TO SOLID TUMORS PNLIP, CETP, NPC1L1 EPHX2 3171/4885FAAH 1988/4885TERT 2358/4885
US-20240100166-A1 NOVEL LIPID FORMULATIONS FOR DELIVERY OF THERAPEUTIC AGENTS PNLIP, NPC1L1, CETP EPHX2 3146/4885FAAH 2156/4885TERT 2551/4885
US-20240182895-A1 NON-LIPOSOMAL SYSTEMS FOR NUCLEIC ACID DELIVERY SNRPE, NPC1L1, LIPA EPHX2 3774/4885FAAH 2035/4885TERT 2828/4885
US-20110117125-A1 COMPOSITIONS AND METHODS FOR THE DELIVERY OF NUCLEIC ACIDS LDLR, SNRPE, SARNP EPHX2 3235/4885FAAH 3989/4885TERT 1679/4885
US-20240050463-A1 THERAPEUTIC COMPOSITIONS AND METHODS FOR TREATING HEPATITIS B HAVCR2, FABP1, HDGF EPHX2 561/4885FAAH 2822/4885TERT 2849/4885
US-11904052-B2 Methods for ameliorating infusion reactions IL2, CD47, IL5 EPHX2 1595/4885FAAH 1650/4885TERT 3039/4885
US-20240148875-A1 NOVEL LIPID FORMULATIONS FOR DELIVERY OF THERAPEUTIC AGENTS PNLIP, NPC1L1, CETP EPHX2 3146/4885FAAH 2156/4885TERT 2551/4885
US-20240035030-A1 NON-LIPOSOMAL SYSTEMS FOR NUCLEIC ACID DELIVERY SNRPE, NPC1L1, LIPA EPHX2 3774/4885FAAH 2035/4885TERT 2828/4885
US-20110201667-A1 COMPOSITIONS AND METHODS FOR SILENCING EBOLA VIRUS GENE EXPRESSION BST2, AGO2, SCARB1 EPHX2 2783/4885FAAH 2338/4885TERT 3295/4885
US-20110195127-A1 COMPOSITIONS AND METHODS FOR SILENCING APOLIPOPROTEIN B APOB, LDLR, APOL1 EPHX2 2492/4885FAAH 2334/4885TERT 3330/4885
US-12016929-B2 Lipid formulations for delivery of therapeutic agents CETP, PNLIP, NPC1L1 EPHX2 3019/4885FAAH 1966/4885TERT 2352/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.