Fumaric Acid

Fumaric Acid

SCHEMBL9795089

NCC(=O)NC1CCC(O[N+](=O)[O-])CC1.O=C(O)C=CC(=O)O

nearest known ligand 0.41

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ATP4AATP4BAXLBTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CHRM2CHRM3CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4FLT3HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3KCNH2KMT2AMAP2K1MAP2K2MEN1MLNRMPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PLK4PPARGRENS1PR1SLC6A2SLC6A3SLC6A4SMOTYK2atpAatpBatpCatpDatpEatpFatpFHatpGpol

The experimentally established mechanism targets of Fumaric Acid. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.36
HTT P42858 1/20 0.36
NPC1 O15118 1/20 0.36
GAA P10253 1/20 0.36
ALDH1A1 P00352 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
BCHE P06276 1/20 0.34
SMYD3 Q9H7B4 3/20 0.33
TMEM97 Q5BJF2 2/20 0.33
NPSR1 Q6W5P4 1/20 0.32
LMNA P02545 2/20 0.31
ATF4 P18848 1/20 0.31
MAPT P10636 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9795195 0.92 ALDH1A1 (0.39) SMN1; SMN2HTTNPC1ALDH1A1L3MBTL1
Fumaric Acid SCHEMBL9795178 0.90 SMYD3 (0.41) POLBSMYD3
Fumaric Acid SCHEMBL9795135 0.83 POLB (0.39) POLBSMN1; SMN2HTTNPC1GAA
SCHEMBL9019551 0.83 POLB (0.64) POLBSMN1; SMN2HTTNPC1GAA
Fumaric Acid SCHEMBL9795498 0.82 TDP1 (0.35) POLBALDH1A1
Fumaric Acid SCHEMBL9795108 0.81 POLB (0.37) POLBSMN1; SMN2HTTNPC1GAA
SCHEMBL9795527 0.80 SMYD3 (0.44) ALDH1A1L3MBTL1SMYD3
SCHEMBL9497980 0.80 SMYD3 (0.44) ALDH1A1L3MBTL1SMYD3
SCHEMBL9497857 0.80 SMYD3 (0.44) ALDH1A1L3MBTL1SMYD3
SCHEMBL9130345 0.78 ALDH1A1 (0.40) SMN1; SMN2HTTNPC1ALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5037849-A For treatment of heart and circulatory diseases BOEHRINGER MANNHEIM GMBH (DE) 1991-08-06 US disclosed