SCHEMBL9824965

SCHEMBL9824965

CN(CC1CCN(CC#N)C1)C1CCCCC1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.33
PGR P06401 1/20 0.31
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30
NOS2 P35228 1/20 0.30
ALDH1A1 P00352 2/20 0.30
HRH4 Q9H3N8 1/20 0.30
PKM P14618 1/20 0.30
ACHE P22303 1/20 0.30
GAA P10253 1/20 0.30
TSHR P16473 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
KDM4E B2RXH2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9823938 0.78 PRMT3 (0.35) HRH3ALDH1A1HRH4PKMACHE
SCHEMBL9824895 0.75 DRD2 (0.34) PGR
SCHEMBL9824823 0.75 MEN1 (0.32) PGR
SCHEMBL9036766 0.73 SIGMAR1 (0.40) HRH3PGRHRH4TSHR
SCHEMBL9824395 0.72 MEN1 (0.34) TSHR
SCHEMBL9824611 0.71 CHRM5 (0.48) HRH3ACHESMN1; SMN2
SCHEMBL9824968 0.71 CXCR4 (0.43) HRH3ACHESMN1; SMN2KDM4E
SCHEMBL27267877 0.71 NOS3 (0.38) HRH3NOS3NOS1NOS2HRH4
SCHEMBL9824712 0.70 MEN1 (0.40) ACHE
SCHEMBL9824002 0.70 OPRM1 (0.32) HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0273239-B1 CONDENSED DIAZEPINONES, PROCESSES FOR THEIR PREPARATION AND MEDICAMENTS CONTAINING THEM Dr. Karl Thomae GmbH (DE) 1991-03-06 EP disclosed
US-4873236-A BRADYCARDIAL AGENTS DR. KARL THOMAE GMBH (DE) 1989-10-10 US disclosed