SCHEMBL9866075

SCHEMBL9866075

CC(COc1ccc(N2N=C3c4cc(F)ccc4CCC3CC2=O)cc1)NCCN1CCCCC1

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.37
ACHE P22303 2/20 0.37
HRH3 Q9Y5N1 6/20 0.35
MCHR1 Q99705 2/20 0.35
DRD2 P14416 2/20 0.34
MAOB P27338 2/20 0.34
MAOA P21397 1/20 0.34
KCNH2 Q12809 2/20 0.34
ESR1 P03372 1/20 0.33
ESR2 Q92731 1/20 0.33
HTR2C P28335 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9602809 0.88 DRD2 (0.34) HTR1AHRH3DRD2MAOBKCNH2
SCHEMBL9602555 0.86 ALDH1A1 (0.34) DRD2MAOB
SCHEMBL9602330 0.85 ESR1 (0.37) HRH3DRD2ESR1ESR2
SCHEMBL9601947 0.82 ADRB1 (0.39)
SCHEMBL9603224 0.82 DRD2 (0.36) HTR1AHRH3DRD2KCNH2HTR2C
SCHEMBL9602515 0.81 ALDH1A1 (0.33) ACHEDRD2
Fumaric Acid SCHEMBL9865911 0.81 KDM4E (0.35) DRD2
SCHEMBL9602850 0.79 DRD2 (0.35) HTR1ADRD2KCNH2ESR1
Hydrochloric Acid SCHEMBL9602310 0.79 S1PR1 (0.33) ACHEDRD2
Fumaric Acid SCHEMBL9602547 0.78 LMNA (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5045541-A Immunodeficiency disorders YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1991-09-03 US disclosed
EP-0351435-A1 FUSED PYRIDAZINE COMPOUNDS AND THEIR MEDICINAL USES Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1990-01-24 EP disclosed