SCHEMBL9954958

SCHEMBL9954958

Nc1nc2ccc(Br)cc2c(=O)n1-c1ccccn1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
KDM4E B2RXH2 1/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
ATM Q13315 1/20 0.46
HTT P42858 1/20 0.44
USP2 O75604 2/20 0.41
MAPT P10636 1/20 0.41
TSHR P16473 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
PTGS2 P35354 1/20 0.41
GABRA1 P14867 1/20 0.41
GABRG2 P18507 1/20 0.41
GABRB3 P28472 1/20 0.41
GABRA5 P31644 1/20 0.41
GABRA3 P34903 1/20 0.41
GABRA2 P47869 1/20 0.41
GABRA6 Q16445 1/20 0.41
IDO1 P14902 1/20 0.41
TDO2 P48775 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24320108 0.85 ALDH1A1 (0.62) ALDH1A1KDM4EMEN1KMT2AATM
SCHEMBL30516932 0.85 ALDH1A1 (0.62) ALDH1A1KDM4EMEN1KMT2AATM
SCHEMBL9953980 0.82 ATM (0.51) ALDH1A1KDM4EMEN1KMT2AATM
SCHEMBL9954930 0.81 POLB (0.58) ALDH1A1KDM4EMEN1KMT2AATM
SCHEMBL2926644 0.81 KMT2A (0.41) MEN1KMT2AHTTUSP2MAPT
SCHEMBL9953464 0.79 ALDH1A1 (0.57) ALDH1A1KDM4EMEN1KMT2AATM
SCHEMBL9954470 0.77 HCAR1 (0.46) ALDH1A1MEN1KMT2AATMHTT
SCHEMBL9954589 0.76 ALOX12 (0.50) ALDH1A1MEN1KMT2AATMMAPT
SCHEMBL24320125 0.75 MEN1 (0.52) ALDH1A1KDM4EMEN1KMT2AATM
SCHEMBL9954662 0.74 PI4KA (0.47) KDM4EMEN1KMT2AATMHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012087938-A1 QUINAZOLINONE DERIVATIVES AS ANTIVIRAL AGENTS GLAXOSMITHKLINE LLC (US) 2012-06-28 WO disclosed